A review on regulation of drug transporters during inflammation / 药学学报
Acta Pharmaceutica Sinica
;
(12): 773-779, 2011.
Article
in Chinese
| WPRIM
| ID: wpr-233057
ABSTRACT
Drug metabolism will change significantly during inflammation, including the reduction of expression and activity of many drug metabolizing enzymes and transporters. Body would release a series of inflammatory cytokines which can regulate drug metabolizing enzymes. Recent studies have revealed that drug transporters are also regulated by the cytokines with obvious species difference. Mechanism studies show that several transcription factors play important roles during the signal pathways of regulation. This review focuses on the progress in the regulation of drug transporters during inflammation.
Full text:
Available
Index:
WPRIM (Western Pacific)
Main subject:
Membrane Transport Proteins
/
Biological Transport
/
Signal Transduction
/
ATP-Binding Cassette Transporters
/
ATP Binding Cassette Transporter, Subfamily B
/
Multidrug Resistance-Associated Proteins
/
Organic Anion Transporters
/
Organic Cation Transport Proteins
/
ATP Binding Cassette Transporter, Subfamily G, Member 2
/
ATP Binding Cassette Transporter, Subfamily B, Member 11
Limits:
Animals
/
Humans
Language:
Chinese
Journal:
Acta Pharmaceutica Sinica
Year:
2011
Type:
Article
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