Advances in the study of affinity selection-ultrafiltration/HPLC-MS / 药学学报
Acta Pharmaceutica Sinica
;
(12): 1084-1088, 2009.
Artículo
en Chino
| WPRIM
| ID: wpr-344053
ABSTRACT
Affinity selection-ultrafiltration/HPLC-MS is the combination of the ultrafiltration and HPLC-MS, mainly used for screening small active molecular substances from combinatorial libraries and natural product extracts, which can bind to solution-phase targets. Besides, it can be used in metabolic screening and characterization of ligand-receptor binding. It is a complement to the traditional methods of screening and identifying drugs. This review describes its principle and application in drug study.
Texto completo:
Disponible
Índice:
WPRIM (Pacífico Occidental)
Asunto principal:
Unión Proteica
/
Espectrometría de Masas
/
Preparaciones Farmacéuticas
/
Ultrafiltración
/
Cromatografía Líquida de Alta Presión
/
Técnicas Químicas Combinatorias
/
Evaluación Preclínica de Medicamentos
/
Bibliotecas de Moléculas Pequeñas
/
Ligandos
/
Metabolismo
Límite:
Humanos
Idioma:
Chino
Revista:
Acta Pharmaceutica Sinica
Año:
2009
Tipo del documento:
Artículo
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