Action of protein phosphatase-1 on Tat-dependent HIV-1 transcription and its related inhibitors / 药学学报
Acta Pharmaceutica Sinica
;
(12): 1343-1347, 2009.
Artículo
en Chino
| WPRIM
| ID: wpr-344074
ABSTRACT
Host cell protein phosphatase-1 (PP1) is an important regulator of human immunodeficiency virus-1 (HIV-1) transcription. PP1 is involved in the regulation of HIV-1 transcription, and dephosphorylates RNA polymerase II C-terminal domain (RNAPII CTD) or CycT1-dependent kinase 9 (CDK9) to increase Tat-dependent HIV-1 transcription. In this review, we discuss the action of PP1 in Tat-induced HIV-1 transcription and related to PP1 inhibitors.
Texto completo:
Disponible
Índice:
WPRIM (Pacífico Occidental)
Asunto principal:
Farmacología
/
Fisiología
/
Piranos
/
Compuestos de Espiro
/
Transcripción Genética
/
Química
/
VIH-1
/
Ácido Ocadaico
/
Fármacos Anti-VIH
/
Inhibidores Enzimáticos
Límite:
Humanos
Idioma:
Chino
Revista:
Acta Pharmaceutica Sinica
Año:
2009
Tipo del documento:
Artículo
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