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Advances in models for predicting drug intestinal permeability / 药学学报
Acta Pharmaceutica Sinica ; (12): 727-734, 2018.
Artículo en Chino | WPRIM | ID: wpr-779928
ABSTRACT
Intestinal permeability is one of key factors determing absorption of oral drug products. It is a big challenge to assess permeability of compounds with high accuracy and high efficacy during research and development process. In this review, the principles, strengths, weaknesses and advances of common intestinal permeability models are summarized, with focus on Ussing chamber and parallel artificial membrane permeability assay. In addition, future trends of permeability models are briefly discussed. This review may provide a reference to accessing permeability of lead compounds.

Texto completo: Disponible Índice: WPRIM (Pacífico Occidental) Tipo de estudio: Estudio pronóstico Idioma: Chino Revista: Acta Pharmaceutica Sinica Año: 2018 Tipo del documento: Artículo

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Texto completo: Disponible Índice: WPRIM (Pacífico Occidental) Tipo de estudio: Estudio pronóstico Idioma: Chino Revista: Acta Pharmaceutica Sinica Año: 2018 Tipo del documento: Artículo