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Study on contribution of main components in Guizhi Fuling capsule based on molecular imprinting technique and activity screening / 中国中药杂志
China Journal of Chinese Materia Medica ; (24): 2420-2427, 2015.
Artigo em Chinês | WPRIM | ID: wpr-337918
ABSTRACT
To clarify the active components in Guizhi Fuling capsule in treatment of intrinsic dysmenorrhea, pelvic inflammation and hysteromyoma, main components were gradually knocked out from the capsules, the effects of knockout capsules on uterine contraction, TNF-α secretion, murine splenocytes (SPL) and hysteromyoma cells proliferation were evaluated, respectively. The inhibition of capsules on uterine contraction was weakened by gradient knockout of paeoniflorin, paeonol, and amygdalin. The suppression of capsulte on TNF-α secretion was reduced by gradient knockout of gallic acid, cinnamaldehyde, pentagalloylglucose, and pachyman. The promotion of SPL cells proliferation was reversed by gradient knockout of gallic acid, paeoniflorin, cinnamaldehyde, quercetin, and pachyman. The depression of capsules on hysteromyoma cells proliferation was attenuated by gradient knockout of paeoniflorin, paeonol, pentagalloylglucose, and albiflorin. In conclusion, the compounds mentioned-above could be the key active basis of Guizhi Fuling capsule in treatment of intrinsic dysmenorrhea, pelvic inflammation and hysteromyoma.
Assuntos
Texto completo: DisponíveL Índice: WPRIM (Pacífico Ocidental) Assunto principal: Cápsulas / Medicamentos de Ervas Chinesas / Química / Fator de Necrose Tumoral alfa / Proliferação de Células / Tratamento Farmacológico / Dismenorreia / Impressão Molecular / Metabolismo / Métodos Tipo de estudo: Estudo diagnóstico / Estudo de rastreamento Limite: Animais / Feminino / Humanos Idioma: Chinês Revista: China Journal of Chinese Materia Medica Ano de publicação: 2015 Tipo de documento: Artigo

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Texto completo: DisponíveL Índice: WPRIM (Pacífico Ocidental) Assunto principal: Cápsulas / Medicamentos de Ervas Chinesas / Química / Fator de Necrose Tumoral alfa / Proliferação de Células / Tratamento Farmacológico / Dismenorreia / Impressão Molecular / Metabolismo / Métodos Tipo de estudo: Estudo diagnóstico / Estudo de rastreamento Limite: Animais / Feminino / Humanos Idioma: Chinês Revista: China Journal of Chinese Materia Medica Ano de publicação: 2015 Tipo de documento: Artigo