Lead compound optimization strategy (6)-improving the plasma stability / 药学学报
Acta Pharmaceutica Sinica
;
(12): 192-201, 2018.
Artigo
em Chinês
| WPRIM
| ID: wpr-779863
ABSTRACT
Plasma stability plays an important role in the druggability of lead compound. Improving the plasma stability of compounds by structural modification can lead to good pharmacokinetic and pharmacodynamics properties. This review provides a summary of varieties of structure modification strategies for improving plasma stability including bioisosterism, increasing steric hindrance, ring closure, scaffold hopping and etc.
Texto completo:
DisponíveL
Índice:
WPRIM (Pacífico Ocidental)
Idioma:
Chinês
Revista:
Acta Pharmaceutica Sinica
Ano de publicação:
2018
Tipo de documento:
Artigo
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