Detalles de la búsqueda
1.
Pharmacological and toxicological evaluation of methyl 4-hydroxy-2H-1,2-benzothiazine-3-carboxylate 1,1-dioxoide against haloperidol induced Parkinson like symptoms in animal model: In-vitro and in-vivo studies.
Toxicol Appl Pharmacol
; 477: 116678, 2023 10 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-37683697
2.
Recent synthetic approaches towards thienothiophenes: a potential template for biologically active compounds.
Mol Divers
; 2023 Apr 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-37095354
3.
A Comprehensive Update of Various Attempts by Medicinal Chemists to Combat COVID-19 through Natural Products.
Molecules
; 28(12)2023 Jun 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-37375415
4.
Recent trends in the chemistry of Sandmeyer reaction: a review.
Mol Divers
; 26(3): 1837-1873, 2022 Jun.
Artículo
en Inglés
| MEDLINE | ID: mdl-34417715
5.
Highly Selective Methodology for Entrapment and Subsequent Removal of Cobalt (II) Ions under Optimized Conditions by Micellar-Enhanced Ultrafiltration.
Molecules
; 27(23)2022 Nov 29.
Artículo
en Inglés
| MEDLINE | ID: mdl-36500426
6.
Synthesis of Novel N-Methylmorpholine-Substituted Benzimidazolium Salts as Potential α-Glucosidase Inhibitors.
Molecules
; 27(18)2022 Sep 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-36144750
7.
Discovery of Novel HCV NS5B polymerase inhibitor, 2-(3,4-dimethyl-5,5-dioxidobenzo[e]pyrazolo[4,3-c][1,2]thiazin-2(4H)-yl)-N-(2-fluorobenzyl)acetamide via molecular docking and experimental approach.
Clin Exp Pharmacol Physiol
; 48(12): 1653-1661, 2021 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-34386985
8.
Discovery of Amide-Functionalized Benzimidazolium Salts as Potent α-Glucosidase Inhibitors.
Molecules
; 26(16)2021 Aug 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-34443347
9.
Synthesis and α-Glucosidase Inhibition Activity of 2-[3-(Benzoyl/4-bromobenzoyl)-4-hydroxy-1,1-dioxido-2H-benzo[e][1,2]thiazin-2-yl]-N-arylacetamides: An In Silico and Biochemical Approach.
Molecules
; 26(10)2021 May 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-34065194
10.
Synthesis and α-glucosidase inhibition studies of norfloxacin-acetanilide hybrids.
Pak J Pharm Sci
; 34(5(Supplementary)): 1909-1915, 2021 Sep.
Artículo
en Inglés
| MEDLINE | ID: mdl-34836859
11.
In-silico modeling and in-vitro studies of 2,1-benzothiazine-2,2-dioxide based hydrazone derivatives as α-glucosidase inhibitors.
Pak J Pharm Sci
; 34(5(Supplementary)): 1951-1955, 2021 Sep.
Artículo
en Inglés
| MEDLINE | ID: mdl-34836865
12.
Synthesis, spectral analysis and biological evaluation of 2-{[(morpholin-4-yl)ethyl]thio}-5-phenyl/aryl-1,3,4-oxadiazole derivatives.
Pak J Pharm Sci
; 34(1(Special)): 441-446, 2021 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-34275792
13.
Development of green methodologies for Heck, Chan-Lam, Stille and Suzuki cross-coupling reactions.
Mol Divers
; 24(3): 821-839, 2020 Aug.
Artículo
en Inglés
| MEDLINE | ID: mdl-31463833
14.
Synthesis, molecular docking and anti-diabetic studies of novel benzimidazole-pyrazoline hybrid molecules.
Pak J Pharm Sci
; 33(2(Supplementary)): 847-854, 2020 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-32863261
15.
Synthesis, characterization and antimicrobial activity of norfloxacin based acetohydrazides.
Pak J Pharm Sci
; 33(2(Supplementary)): 855-860, 2020 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-32863262
16.
Benzothiazine based acetohydrazides and acetamides as anticancer agents.
Pak J Pharm Sci
; 32(6(Supplementary)): 2795-2800, 2019 Nov.
Artículo
en Inglés
| MEDLINE | ID: mdl-32024616
17.
Alpha-glucosidase inhibition and molecular docking studies of 1,2-benzothiazine 1,1-dioxide based carbohydrazides.
Pak J Pharm Sci
; 32(6(Supplementary)): 2829-2834, 2019 Nov.
Artículo
en Inglés
| MEDLINE | ID: mdl-32024621
18.
Design, synthesis, in-silico study and anticancer potential of novel n-4- piperazinyl-ciprofloxacin-aniline hybrids.
Pak J Pharm Sci
; 32(5(Supplementary)): 2215-2222, 2019 Sep.
Artículo
en Inglés
| MEDLINE | ID: mdl-31894047
19.
Malic enzyme 2 as a potential therapeutic drug target for cancer.
IUBMB Life
; 70(11): 1076-1083, 2018 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-30160039
20.
Synthesis, characterization, monoamine oxidase inhibition, molecular docking and dynamic simulations of novel 2,1-benzothiazine-2,2-dioxide derivatives.
Bioorg Chem
; 80: 498-510, 2018 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-29996111