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1.
Pharmacological Characterization of the Microsomal Prostaglandin E2 Synthase-1 Inhibitor AF3485 In Vitro and In Vivo.
Front Pharmacol
; 11: 374, 2020.
Artículo
en Inglés
| MEDLINE | ID: mdl-32317963
2.
The anti-inflammatory agent bindarit acts as a modulator of fatty acid-binding protein 4 in human monocytic cells.
Sci Rep
; 9(1): 15155, 2019 10 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-31641194
3.
Identification of potent triazolylpyridine nicotinamide phosphoribosyltransferase (NAMPT) inhibitors bearing a 1,2,3-triazole tail group.
Eur J Med Chem
; 181: 111576, 2019 Nov 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-31400709
4.
Targeting Serotonin 2A and Adrenergic α1 Receptors for Ocular Antihypertensive Agents: Discovery of 3,4-Dihydropyrazino[1,2-b]indazol-1(2H)-one Derivatives.
ChemMedChem
; 13(15): 1597-1607, 2018 08 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-29873449
5.
Identification of Novel Triazole-Based Nicotinamide Phosphoribosyltransferase (NAMPT) Inhibitors Endowed with Antiproliferative and Antiinflammatory Activity.
J Med Chem
; 60(5): 1768-1792, 2017 03 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-28165742
6.
Hit Optimization of 5-Substituted-N-(piperidin-4-ylmethyl)-1H-indazole-3-carboxamides: Potent Glycogen Synthase Kinase-3 (GSK-3) Inhibitors with in Vivo Activity in Model of Mood Disorders.
J Med Chem
; 58(22): 8920-37, 2015 Nov 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-26486317
7.
Pharmacological inhibition of microsomal prostaglandin E synthase-1 suppresses epidermal growth factor receptor-mediated tumor growth and angiogenesis.
PLoS One
; 7(7): e40576, 2012.
Artículo
en Inglés
| MEDLINE | ID: mdl-22815767
8.
Discovery and pharmacological profile of new 1H-indazole-3-carboxamide and 2H-pyrrolo[3,4-c]quinoline derivatives as selective serotonin 4 receptor ligands.
J Med Chem
; 55(22): 9446-66, 2012 Nov 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-23043420
9.
Effects of AF3442 [N-(9-ethyl-9H-carbazol-3-yl)-2-(trifluoromethyl)benzamide], a novel inhibitor of human microsomal prostaglandin E synthase-1, on prostanoid biosynthesis in human monocytes in vitro.
Biochem Pharmacol
; 79(7): 974-81, 2010 Apr 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-19925781
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