Detalles de la búsqueda
1.
Multiplexed cellular profiling identifies an organoselenium compound as an inhibitor of CRM1-mediated nuclear export.
Traffic
; 23(12): 587-599, 2022 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-36353954
2.
Generation and characterisation of an Arabidopsis thaliana f3h/fls1/ans triple mutant that accumulates eriodictyol derivatives.
BMC Plant Biol
; 24(1): 99, 2024 Feb 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-38331743
3.
Sulfonamide-incorporated bis(α-aminophosphonates) as promising carbonic anhydrase inhibitors: Design, synthesis, biological evaluation, and X-ray crystallographic studies.
Arch Pharm (Weinheim)
; : e2400038, 2024 Mar 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-38498884
4.
Design, synthesis, and biological evaluation of 3-benzenesulfonamide-linked 3-hydrazinoisatin derivatives as carbonic anhydrase inhibitors.
Arch Pharm (Weinheim)
; 357(6): e2300718, 2024 Jun.
Artículo
en Inglés
| MEDLINE | ID: mdl-38466120
5.
Identification of 3-(5-cyano-6-oxo-pyridin-2-yl)benzenesulfonamides as novel anticancer agents endowed with EGFR inhibitory activity.
Arch Pharm (Weinheim)
; 357(1): e2300449, 2024 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-37828544
6.
Leveraging SARS-CoV-2 Main Protease (Mpro) for COVID-19 Mitigation with Selenium-Based Inhibitors.
Int J Mol Sci
; 25(2)2024 Jan 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-38256046
7.
Mono- and three-tailed sugar and iminosugar decorated benzenesulfonamide carbonic anhydrase inhibitors.
Org Biomol Chem
; 21(21): 4491-4503, 2023 05 31.
Artículo
en Inglés
| MEDLINE | ID: mdl-37198937
8.
Substituted furan sulfonamides as carbonic anhydrase inhibitors: Synthesis, biological and in silico studies.
Bioorg Chem
; 138: 106621, 2023 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-37257407
9.
Schiff bases as linker in the development of quinoline-sulfonamide hybrids as selective cancer-associated carbonic anhydrase isoforms IX/XII inhibitors: A new regioisomerism tactic.
Bioorg Chem
; 131: 106309, 2023 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-36502567
10.
Click chemistry approaches for developing carbonic anhydrase inhibitors and their applications.
J Enzyme Inhib Med Chem
; 38(1): 2166503, 2023 Jan 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-36637011
11.
Diversely N-substituted benzenesulfonamides dissimilarly bind to human carbonic anhydrases: crystallographic investigations of N-nitrosulfonamides.
J Enzyme Inhib Med Chem
; 38(1): 2178430, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36798036
12.
Cloning, characterization, and inhibition of the novel ß-carbonic anhydrase from parasitic blood fluke, Schistosoma mansoni.
J Enzyme Inhib Med Chem
; 38(1): 2184299, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36856011
13.
Synthesis and biological evaluation of new 3-substituted coumarin derivatives as selective inhibitors of human carbonic anhydrase IX and XII.
J Enzyme Inhib Med Chem
; 38(1): 2185760, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36876597
14.
Selenium-analogs based on natural sources as cancer-associated carbonic anhydrase isoforms IX and XII inhibitors.
J Enzyme Inhib Med Chem
; 38(1): 2191165, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36938694
15.
Benzenesulfonamide derivatives as Vibrio cholerae carbonic anhydrases inhibitors: a computational-aided insight in the structural rigidity-activity relationships.
J Enzyme Inhib Med Chem
; 38(1): 2201402, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-37073528
16.
2H-chromene and 7H-furo-chromene derivatives selectively inhibit tumour associated human carbonic anhydrase IX and XII isoforms.
J Enzyme Inhib Med Chem
; 38(1): 2270183, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-37870190
17.
Discovery of sulfonamide-tethered isatin derivatives as novel anticancer agents and VEGFR-2 inhibitors.
J Enzyme Inhib Med Chem
; 38(1): 2203389, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-37122176
18.
Structure-guided identification of a selective sulfonamide-based inhibitor targeting the human carbonic anhydrase VA isoform.
Arch Pharm (Weinheim)
; 356(1): e2200383, 2023 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-36250310
19.
Benzenesulfonamides with trisubstituted triazole motif as selective carbonic anhydrase I, II, IV, and IX inhibitors.
Arch Pharm (Weinheim)
; 356(1): e2200391, 2023 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-36316236
20.
Tail approach synthesis of triazolylthiazolotriazole bearing benzenesulfonamides as carbonic anhydrase inhibitors capable of inducing apoptosis.
Arch Pharm (Weinheim)
; 356(2): e2200439, 2023 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-36344431