Detalles de la búsqueda
1.
Design, in silico study, synthesis and evaluation of hybrid pyrazole substituted 1,3,5-triazine derivatives for antimalarial activity.
Exp Parasitol
; 261: 108767, 2024 Jun.
Artículo
en Inglés
| MEDLINE | ID: mdl-38679125
2.
In silico screening, synthesis, and antimalarial evaluation of PABA substituted 1,3,5-triazine derivatives as Pf-DHFR inhibitors.
Exp Parasitol
; 250: 108546, 2023 Jul.
Artículo
en Inglés
| MEDLINE | ID: mdl-37196703
3.
Pharmacoinformatics-based identification of transmembrane protease serine-2 inhibitors from Morus Alba as SARS-CoV-2 cell entry inhibitors.
Mol Divers
; 26(1): 265-278, 2022 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-33786727
4.
Facile synthesis, antimicrobial and antiviral evaluation of novel substituted phenyl 1,3-thiazolidin-4-one sulfonyl derivatives.
Bioorg Chem
; 114: 105153, 2021 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-34328851
5.
Synthesis and biological evaluation of substituted phenyl azetidine-2-one sulphonyl derivatives as potential antimicrobial and antiviral agents.
Bioorg Chem
; 104: 104320, 2020 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-33142428
6.
Acute and sub-chronic toxicity studies of Benincasa hispida (Thunb.) cogniaux fruit extract in rodents.
Regul Toxicol Pharmacol
; 118: 104785, 2020 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-32976857
7.
Design, synthesis and antimalarial screening of some hybrid 4-aminoquinoline-triazine derivatives against pf-DHFR-TS.
Exp Parasitol
; 163: 38-45, 2016 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-26821296
8.
Synthesis, antimalarial activity and molecular docking of hybrid 4-aminoquinoline-1,3,5-triazine derivatives.
Exp Parasitol
; 157: 59-67, 2015 Oct.
Artículo
en Inglés
| MEDLINE | ID: mdl-26164360
9.
Structure-guided discovery of 1,3,5-triazine-pyrazole conjugates as antibacterial and antibiofilm agent against pathogens causing human diseases with favorable metabolic fate.
Bioorg Med Chem Lett
; 24(15): 3321-5, 2014 Aug 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-24961639
10.
A Review on Synthetic Thiazole Derivatives as an Antimalarial Agent.
Curr Drug Discov Technol
; 2024 Jan 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-38279721
11.
Physicochemical characterization and in vitro dissolution studies of solid dispersions of ketoprofen with PVP K30 and d-mannitol.
Saudi Pharm J
; 21(1): 77-84, 2013 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-24109206
12.
Discovery of imeglimin-inspired novel 1,3,5-triazine derivatives as antidiabetic agents in streptozotocin-induced diabetes in Wistar rats via inhibition of DPP-4.
RSC Med Chem
; 14(8): 1512-1536, 2023 Aug 16.
Artículo
en Inglés
| MEDLINE | ID: mdl-37593577
13.
Discovery of novel 1,3,5-triazine derivatives as an antidiabetic agent in Wistar rats via inhibition of DPP-4.
Future Med Chem
; 15(10): 829-852, 2023 May.
Artículo
en Inglés
| MEDLINE | ID: mdl-37307171
14.
Hybrid PABA-glutamic acid conjugated 1,3,5-triazine derivatives: Design, synthesis, and antimalarial activity screening targeting Plasmodium falciparum dihydro folate reductase enzyme.
Chem Biol Drug Des
; 102(6): 1336-1352, 2023 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-37783571
15.
Molecular docking and antimalarial evaluation of hybrid para-aminobenzoic acid 1,3,5 triazine derivatives via inhibition of Pf-DHFR.
J Biomol Struct Dyn
; 41(24): 15520-15534, 2023.
Artículo
en Inglés
| MEDLINE | ID: mdl-37154740
16.
Antimalarial evaluation and docking studies of hybrid phenylthiazolyl-1,3,5-triazine derivatives: a novel and potential antifolate lead for Pf-DHFR-TS inhibition.
Exp Parasitol
; 130(3): 292-9, 2012 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-22233734
17.
Synthesis, SAR and antibacterial activity of hybrid chloro, dichloro-phenylthiazolyl-s-triazines.
Saudi Pharm J
; 20(1): 35-43, 2012 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-23960775
18.
A Review Of Preclinical Tools To Validate Anti-Diarrheal Agents.
Curr Rev Clin Exp Pharmacol
; 2022 Nov 21.
Artículo
en Inglés
| MEDLINE | ID: mdl-36411576
19.
Molecular insights into a mechanism of resveratrol action using hybrid computational docking/CoMFA and machine learning approach.
J Biomol Struct Dyn
; 40(18): 8286-8300, 2022 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-33829956
20.
Molecular docking and antimalarial evaluation of novel N-(4-aminobenzoyl)-l-glutamic acid conjugated 1,3,5-triazine derivatives as Pf-DHFR inhibitors.
3 Biotech
; 12(12): 347, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36386564