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1.
Discovery and Optimization of Pyridazinones as PI3Kδ Selective Inhibitors for Administration by Inhalation.
J Med Chem
; 2024 Jun 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-38907711
2.
1H NMR discrimination of CHF4226.01 diastereoisomers in DMSO-d6.
Magn Reson Chem
; 47(7): 551-61, 2009 Jul.
Artículo
en Inglés
| MEDLINE | ID: mdl-19373771
3.
Atropisomerism and Conformational Equilibria: Impact on PI3Kδ Inhibition of 2-((6-Amino-9H-purin-9-yl)methyl)-5-methyl-3-(o-tolyl)quinazolin-4(3H)-one (IC87114) and Its Conformationally Restricted Analogs.
J Med Chem
; 60(10): 4304-4315, 2017 05 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-28489362
4.
Discovery and Optimization of Thiazolidinyl and Pyrrolidinyl Derivatives as Inhaled PDE4 Inhibitors for Respiratory Diseases.
J Med Chem
; 60(24): 10026-10046, 2017 12 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-29200281
5.
Zinc complexes with cyclic derivatives of alpha-ketoglutaric acid thiosemicarbazone: Synthesis, X-ray structures and DNA interactions.
J Inorg Biochem
; 99(7): 1504-13, 2005 Jul.
Artículo
en Inglés
| MEDLINE | ID: mdl-15927259
6.
Synthesis, characterization and X-ray structures of new antiproliferative and proapoptotic natural aldehyde thiosemicarbazones and their nickel(II) and copper(II) complexes.
J Inorg Biochem
; 90(3-4): 113-26, 2002 Jun 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-12031803
7.
Novel class of benzoic acid ester derivatives as potent PDE4 inhibitors for inhaled administration in the treatment of respiratory diseases.
J Med Chem
; 57(3): 793-816, 2014 Feb 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-24400806
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