Detalles de la búsqueda
1.
PHA-680626 Is an Effective Inhibitor of the Interaction between Aurora-A and N-Myc.
Int J Mol Sci
; 22(23)2021 Dec 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-34884931
2.
Single-Nucleotide Polymorphism of PPARγ, a Protein at the Crossroads of Physiological and Pathological Processes.
Int J Mol Sci
; 18(2)2017 Feb 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-28208577
3.
Catechol-based matrix metalloproteinase inhibitors with additional antioxidative activity.
J Enzyme Inhib Med Chem
; 31(sup4): 25-37, 2016.
Artículo
en Inglés
| MEDLINE | ID: mdl-27556138
4.
Structural basis of the transactivation deficiency of the human PPARγ F360L mutant associated with familial partial lipodystrophy.
Acta Crystallogr D Biol Crystallogr
; 70(Pt 7): 1965-76, 2014 Jul.
Artículo
en Inglés
| MEDLINE | ID: mdl-25004973
5.
A chemical modification of a peroxisome proliferator-activated receptor pan agonist produced a shift to a new dual alpha/gamma partial agonist endowed with mitochondrial pyruvate carrier inhibition and antidiabetic properties.
Eur J Med Chem
; 275: 116567, 2024 Jun 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-38865743
6.
Electrochemical and Structural Characterization of Lanthanum-Doped Hydroxyapatite: A Promising Material for Sensing Applications.
Materials (Basel)
; 16(13)2023 Jun 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-37444835
7.
Biological Screening and Crystallographic Studies of Hydroxy γ-Lactone Derivatives to Investigate PPARγ Phosphorylation Inhibition.
Biomolecules
; 13(4)2023 04 19.
Artículo
en Inglés
| MEDLINE | ID: mdl-37189440
8.
Novel N-(Heterocyclylphenyl)benzensulfonamide Sharing an Unreported Binding Site with T-Cell Factor 4 at the ß-Catenin Armadillo Repeats Domain as an Anticancer Agent.
ACS Pharmacol Transl Sci
; 6(7): 1087-1103, 2023 Jul 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-37470018
9.
Cytosolic localization and in vitro assembly of human de novo thymidylate synthesis complex.
FEBS J
; 289(6): 1625-1649, 2022 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-34694685
10.
Discovery of Novel Chemical Series of OXA-48 ß-Lactamase Inhibitors by High-Throughput Screening.
Pharmaceuticals (Basel)
; 14(7)2021 Jun 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-34202402
11.
Bone-Seeking Matrix Metalloproteinase Inhibitors for the Treatment of Skeletal Malignancy.
Pharmaceuticals (Basel)
; 13(6)2020 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-32492898
12.
A Novel N-Substituted Valine Derivative with Unique Peroxisome Proliferator-Activated Receptor γ Binding Properties and Biological Activities.
J Med Chem
; 63(21): 13124-13139, 2020 11 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-33142057
13.
Insights into PPARγ Phosphorylation and Its Inhibition Mechanism.
J Med Chem
; 63(9): 4811-4823, 2020 05 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-32239932
14.
Surface Plasmon Resonance as a Tool for Ligand Binding Investigation of Engineered GPR17 Receptor, a G Protein Coupled Receptor Involved in Myelination.
Front Chem
; 7: 910, 2019.
Artículo
en Inglés
| MEDLINE | ID: mdl-31998697
15.
Identification of the First PPARα/γ Dual Agonist Able To Bind to Canonical and Alternative Sites of PPARγ and To Inhibit Its Cdk5-Mediated Phosphorylation.
J Med Chem
; 61(18): 8282-8298, 2018 09 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-30199253
16.
Betulinic acid is a PPARγ antagonist that improves glucose uptake, promotes osteogenesis and inhibits adipogenesis.
Sci Rep
; 7(1): 5777, 2017 07 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-28720829
17.
Screening of saponins and sapogenins from Medicago species as potential PPARγ agonists and X-ray structure of the complex PPARγ/caulophyllogenin.
Sci Rep
; 6: 27658, 2016 06 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-27283034
18.
Structural basis for PPAR partial or full activation revealed by a novel ligand binding mode.
Sci Rep
; 6: 34792, 2016 10 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-27708429
19.
On the metabolically active form of metaglidasen: improved synthesis and investigation of its peculiar activity on peroxisome proliferator-activated receptors and skeletal muscles.
ChemMedChem
; 10(3): 555-65, 2015 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-25641779
Resultados
1 -
19
de 19
1
Próxima >
>>