Detalles de la búsqueda
1.
Design, synthesis, and biological evaluation of benzo[d]imidazole-2-carboxamides as new anti-TB agents.
Bioorg Chem
; 107: 104538, 2021 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-33349456
2.
Benzimidazoquinazolines as new potent anti-TB chemotypes: Design, synthesis, and biological evaluation.
Bioorg Chem
; 99: 103774, 2020 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-32224336
3.
An unprecedented intramolecular to intermolecular mechanistic switch in 1,1-diaminoazines leading to differential product formation during the I2-induced tandem oxidative transformation.
Org Biomol Chem
; 17(16): 4129-4138, 2019 04 17.
Artículo
en Inglés
| MEDLINE | ID: mdl-30969300
4.
α-Sulfonamidophosphonates as new anti-mycobacterial chemotypes: Design, development of synthetic methodology, and biological evaluation.
Bioorg Chem
; 82: 246-252, 2019 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-30391855
5.
Can Remote N-Heterocyclic Carbenes Coordinate with Main Group Elements? Synthesis, Structure, and Quantum Chemical Analysis of N+ -Centered Complexes.
Chemistry
; 24(24): 6418-6425, 2018 Apr 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-29504658
6.
Cross-Dehydrogenative Coupling of Heterocyclic Scaffolds with Unfunctionalized Aroyl Surrogates by Palladium(II) Catalyzed C(sp2)-H Aroylation through Organocatalytic Dioxygen Activation.
J Org Chem
; 82(7): 3767-3780, 2017 04 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-28299930
7.
Rationalization of Benzazole-2-carboxylate versus Benzazine-3-one/Benzazine-2,3-dione Selectivity Switch during Cyclocondensation of 2-Aminothiophenols/Phenols/Anilines with 1,2-Biselectrophiles in Aqueous Medium.
J Org Chem
; 82(19): 10077-10091, 2017 10 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-28846411
8.
Design, Synthesis, and Structural Analysis of Divalent N(I) Compounds and Identification of a New Electron-Donating Ligand.
Chemistry
; 22(3): 1088-96, 2016 Jan 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-26615987
9.
Azine-Hydrazone Tautomerism of Guanylhydrazones: Evidence for the Preference Toward the Azine Tautomer.
J Org Chem
; 81(17): 7574-7583, 2016 Sep 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-27494613
10.
Design, development of new synthetic methodology, and biological evaluation of substituted quinolines as new anti-tubercular leads.
Bioorg Med Chem Lett
; 26(24): 5960-5966, 2016 12 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-27839684
11.
Synthesis, biological evaluation and structure-activity relationship of 2-styrylquinazolones as anti-tubercular agents.
Bioorg Med Chem Lett
; 26(11): 2663-9, 2016 06 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-27095514
12.
Design and synthesis of guanylthiourea derivatives as potential inhibitors of Plasmodium falciparum dihydrofolate reductase enzyme.
Bioorg Med Chem Lett
; 24(2): 613-7, 2014 Jan 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-24361001
13.
Hydrogen-bond-driven electrophilic activation for selectivity control: scope and limitations of fluorous alcohol-promoted selective formation of 1,2-disubstituted benzimidazoles and mechanistic insight for rationale of selectivity.
J Org Chem
; 77(22): 10158-67, 2012 Nov 16.
Artículo
en Inglés
| MEDLINE | ID: mdl-23067292
14.
Lack of correlation between catalytic efficiency and basicity of amines during the reaction of aryl methyl ketones with DMF-DMA: an unprecedented supramolecular domino catalysis.
Org Biomol Chem
; 10(2): 281-6, 2012 Jan 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-22057389
15.
Domino synthesis of functionalized pyridine carboxylates under gallium catalysis: Unravelling the reaction pathway and the role of the nitrogen source counter anion.
Chem Asian J
; 17(15): e202200304, 2022 Aug 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-35608137
16.
Benzo[d]thiazole-2-carboxamides as new antituberculosis chemotypes inhibiting mycobacterial ATP phosphoribosyl transferase.
Future Med Chem
; 14(24): 1847-1864, 2022 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-36444737
17.
Bacterial FtsZ inhibition by benzo[d]imidazole-2-carboxamide derivative with anti-TB activity.
Future Med Chem
; 14(19): 1361-1373, 2022 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-36103222
18.
Zinc tetrafluoroborate hydrate as a mild catalyst for epoxide ring opening with amines: scope and limitations of metal tetrafluoroborates and applications in the synthesis of antihypertensive drugs (RS)/(R)/(S)-metoprolols.
J Org Chem
; 76(21): 8768-80, 2011 Nov 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-21899254
19.
Nonsolvent application of ionic liquids: organo-catalysis by 1-alkyl-3-methylimidazolium cation based room-temperature ionic liquids for chemoselective N-tert-butyloxycarbonylation of amines and the influence of the C-2 hydrogen on catalytic efficiency.
J Org Chem
; 76(17): 7132-40, 2011 Sep 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-21774556
20.
Ruthenium (II) Catalyzed C(sp2 )-H Bond Alkenylation of 2-Arylbenzo[d]oxazole and 2-Arylbenzo[d]thiazole with Unactivated Olefins.
Chem Asian J
; 16(1): 87-96, 2021 Jan 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-33230945