Detalles de la búsqueda
1.
Synthesis, kinetic studies and in-silico investigations of novel quinolinyl-iminothiazolines as alkaline phosphatase inhibitors.
J Enzyme Inhib Med Chem
; 38(1): 2163394, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36629454
2.
Investigation of Newly Synthesized Bis-Acyl-Thiourea Derivatives of 4-Nitrobenzene-1,2-Diamine for Their DNA Binding, Urease Inhibition, and Anti-Brain-Tumor Activities.
Molecules
; 28(6)2023 Mar 16.
Artículo
en Inglés
| MEDLINE | ID: mdl-36985680
3.
Design, synthesis, biochemical and in silico characterization of novel naphthalene-thiourea conjugates as potential and selective inhibitors of alkaline phosphatase.
Med Chem Res
; 32(6): 1077-1086, 2023.
Artículo
en Inglés
| MEDLINE | ID: mdl-37305207
4.
Azomethine-clubbed thiazoles as human tissue non-specific alkaline phosphatase (h-TNAP) and intestinal alkaline phosphatase (h-IAP) Inhibitors: kinetics and molecular docking studies.
Mol Divers
; 26(6): 3241-3254, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-35083622
5.
Analysis of 1-Aroyl-3-[3-chloro-2-methylphenyl] Thiourea Hybrids as Potent Urease Inhibitors: Synthesis, Biochemical Evaluation and Computational Approach.
Int J Mol Sci
; 23(19)2022 Oct 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-36232944
6.
Acetophenone-Based 3,4-Dihydropyrimidine-2(1H)-Thione as Potential Inhibitor of Tyrosinase and Ribonucleotide Reductase: Facile Synthesis, Crystal Structure, In-Vitro and In-Silico Investigations.
Int J Mol Sci
; 23(21)2022 Oct 29.
Artículo
en Inglés
| MEDLINE | ID: mdl-36361953
7.
Synthesis, Biological Evaluation, and Molecular Dynamics of Carbothioamides Derivatives as Carbonic Anhydrase II and 15-Lipoxygenase Inhibitors.
Molecules
; 27(24)2022 Dec 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-36557863
8.
Investigations on Anticancer Potentials by DNA Binding and Cytotoxicity Studies for Newly Synthesized and Characterized Imidazolidine and Thiazolidine-Based Isatin Derivatives.
Molecules
; 27(2)2022 Jan 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-35056668
9.
Exploring 2-Tetradecanoylimino-3-aryl-4-methyl-1,3-thiazolines Derivatives as Alkaline Phosphatase Inhibitors: Biochemical Evaluation and Computational Analysis.
Molecules
; 27(19)2022 Oct 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-36235300
10.
Hydrazine clubbed 1,3-thiazoles as potent urease inhibitors: design, synthesis and molecular docking studies.
Mol Divers
; 25(2): 1-13, 2021 May.
Artículo
en Inglés
| MEDLINE | ID: mdl-32095975
11.
Effect of organic solvents on solvatochromic, fluorescence, and electrochemical properties of synthesized thiazolylcoumarin derivatives.
Luminescence
; 36(5): 1189-1197, 2021 Aug.
Artículo
en Inglés
| MEDLINE | ID: mdl-33759314
12.
Exploring Amantadine Derivatives as Urease Inhibitors: Molecular Docking and Structure-Activity Relationship (SAR) Studies.
Molecules
; 26(23)2021 Nov 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-34885728
13.
Donor-Pi-Acceptor Fluorene Conjugates, Based on Chalcone and Pyrimidine Derivatives: an Insight into Structure-Property Relationship, Photophysical and Electrochemical Properties.
J Fluoresc
; 30(2): 419-426, 2020 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-32095970
14.
Aroylthiourea derivatives of ciprofloxacin drug as DNA binder: Theoretical, spectroscopic and electrochemical studies along with cytotoxicity assessment.
Arch Biochem Biophys
; 666: 83-98, 2019 05 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-30951683
15.
Design, synthesis and biological evaluation of trinary benzocoumarin-thiazoles-azomethines derivatives as effective and selective inhibitors of alkaline phosphatase.
Bioorg Chem
; 91: 103137, 2019 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-31400554
16.
Synthesis of sulfonamide, amide and amine hybrid pharmacophore, an entry of new class of carbonic anhydrase II inhibitors and evaluation of chemo-informatics and binding analysis.
Bioorg Chem
; 86: 624-630, 2019 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-30807935
17.
One-pot four-component synthesis of thiazolidin-2-imines using CuI/ZnII dual catalysis: A new class of acetylcholinesterase inhibitors.
Bioorg Chem
; 84: 518-528, 2019 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-30610971
18.
Synthesis, molecular docking and kinetic studies of novel quinolinyl based acyl thioureas as mushroom tyrosinase inhibitors and free radical scavengers.
Bioorg Chem
; 90: 103063, 2019 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-31220666
19.
Investigation on the effect of alkyl chain linked mono-thioureas as Jack bean urease inhibitors, SAR, pharmacokinetics ADMET parameters and molecular docking studies.
Bioorg Chem
; 86: 473-481, 2019 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-30772648
20.
Drug-1,3,4-Thiadiazole Conjugates as Novel Mixed-Type Inhibitors of Acetylcholinesterase: Synthesis, Molecular Docking, Pharmacokinetics, and ADMET Evaluation.
Molecules
; 24(5)2019 Feb 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-30823444