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Mitogen-activated protein kinase-activated protein kinase 2 (MAPKAP-K2) as an antiinflammatory target: discovery and in vivo activity of selective pyrazolo[1,5-a]pyrimidine inhibitors using a focused library and structure-based optimization approach.
J Med Chem
; 55(15): 6700-15, 2012 Aug 09.
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| MEDLINE | ID: mdl-22746295
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