Detalles de la búsqueda
1.
Probes for narcotic receptor mediated phenomena. 47. Novel C4a- and N-substituted-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-6-ols.
Bioorg Med Chem
; 21(11): 3298-309, 2013 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-23618710
2.
An efficient synthesis of 3-OBn-6ß,14-epoxy-bridged opiates from naltrexone and identification of a related dual MOR inverse agonist/KOR agonist.
Bioorg Med Chem Lett
; 22(22): 6801-5, 2012 Nov 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-22771010
3.
Semisynthetic neoclerodanes as kappa opioid receptor probes.
Bioorg Med Chem
; 20(9): 3100-10, 2012 May 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-22464684
4.
Probes for narcotic receptor mediated phenomena. 43. Synthesis of the ortho-a and para-a, and improved synthesis and optical resolution of the ortho-b and para-b oxide-bridged phenylmorphans: compounds with moderate to low opioid-receptor affinity.
Bioorg Med Chem
; 19(14): 4330-7, 2011 Jul 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-21684752
5.
Probes for narcotic receptor mediated phenomena. Part 42: synthesis and in vitro pharmacological characterization of the N-methyl and N-phenethyl analogues of the racemic ortho-c and para-c oxide-bridged phenylmorphans.
Bioorg Med Chem
; 19(11): 3434-43, 2011 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-21570305
6.
Opioid receptor probes derived from cycloaddition of the hallucinogen natural product salvinorin A.
J Nat Prod
; 74(4): 718-26, 2011 Apr 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-21338114
7.
Identification of a novel "almost neutral" micro-opioid receptor antagonist in CHO cells expressing the cloned human mu-opioid receptor.
Synapse
; 64(4): 280-8, 2010 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-19953652
8.
Probes for narcotic receptor mediated phenomena. 40. N-substituted cis-4a-ethyl-1,2,3,4,4a,9a-hexahydrobenzofuro[2,3-c]pyridin-8-ols.
Bioorg Med Chem
; 18(1): 91-9, 2010 Jan 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-20005115
9.
Studies of the biogenic amine transporters. 13. Identification of "agonist" and "antagonist" allosteric modulators of amphetamine-induced dopamine release.
J Pharmacol Exp Ther
; 329(2): 718-28, 2009 May.
Artículo
en Inglés
| MEDLINE | ID: mdl-19244097
10.
Design, synthesis, and characterization of 6beta-naltrexol analogs, and their selectivity for in vitro opioid receptor subtypes.
Bioorg Med Chem Lett
; 19(10): 2811-4, 2009 May 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-19364645
11.
Synthetic studies of neoclerodane diterpenes from Salvia divinorum: role of the furan in affinity for opioid receptors.
Org Biomol Chem
; 7(18): 3748-56, 2009 Sep 21.
Artículo
en Inglés
| MEDLINE | ID: mdl-19707679
12.
Synthetic studies on neoclerodane diterpenes from Salvia splendens: oxidative modifications of ring A.
Tetrahedron
; 65(8): 1708-1715, 2009 Feb 21.
Artículo
en Inglés
| MEDLINE | ID: mdl-21544261
13.
Studies of the biogenic amine transporters. 12. Identification of novel partial inhibitors of amphetamine-induced dopamine release.
J Pharmacol Exp Ther
; 326(1): 286-95, 2008 Jul.
Artículo
en Inglés
| MEDLINE | ID: mdl-18441249
14.
Design and synthesis of 2- and 3-substituted-3-phenylpropyl analogs of 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine and 1-[2-(diphenylmethoxy)ethyl]-4-(3-phenylpropyl)piperazine: role of amino, fluoro, hydroxyl, methoxyl, methyl, methylene, and oxo substituents on affinity for the dopamine and serotonin transporters.
J Med Chem
; 51(9): 2795-806, 2008 May 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-18393401
15.
Herkinorin analogues with differential beta-arrestin-2 interactions.
J Med Chem
; 51(8): 2421-31, 2008 Apr 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-18380425
16.
Evidence for a mu-delta opioid receptor complex in CHO cells co-expressing mu and delta opioid peptide receptors.
Peptides
; 29(8): 1424-31, 2008 Aug.
Artículo
en Inglés
| MEDLINE | ID: mdl-18472184
17.
Synthesis and pharmacological effects of the enantiomers of the N-phenethyl analogues of the ortho and para e- and f-oxide-bridged phenylmorphans.
Org Biomol Chem
; 6(16): 2868-83, 2008 Aug 21.
Artículo
en Inglés
| MEDLINE | ID: mdl-18688479
18.
Synthetic studies of neoclerodane diterpenoids from Salvia splendens and evaluation of Opioid Receptor affinity.
Tetrahedron
; 64(43): 10041-10048, 2008 Dec 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-20027203
19.
Synthetic studies of neoclerodane diterpenes from Salvia divinorum: preparation and opioid receptor activity of salvinicin analogues.
J Med Chem
; 50(15): 3596-603, 2007 Jul 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-17580847
20.
Probes for narcotic receptor mediated phenomena. 34. Synthesis and structure-activity relationships of a potent mu-agonist delta-antagonist and an exceedingly potent antinociceptive in the enantiomeric C9-substituted 5-(3-hydroxyphenyl)-N-phenylethylmorphan series.
J Med Chem
; 50(16): 3765-76, 2007 Aug 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-17625813