Detalles de la búsqueda
1.
Synthesis, In Silico and Kinetics Evaluation of N-(ß-d-glucopyranosyl)-2-arylimidazole-4(5)-carboxamides and N-(ß-d-glucopyranosyl)-4(5)-arylimidazole-2-carboxamides as Glycogen Phosphorylase Inhibitors.
Int J Mol Sci
; 25(9)2024 Apr 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-38731811
2.
Design and Synthesis of 3-(ß-d-Glucopyranosyl)-4-amino/4-guanidino Pyrazole Derivatives and Analysis of Their Glycogen Phosphorylase Inhibitory Potential.
Molecules
; 28(7)2023 Mar 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-37049768
3.
Stretch-Induced Down-Regulation of HCN2 Suppresses Contractile Activity.
Molecules
; 28(11)2023 May 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-37298834
4.
Mechanosensing in the Physiology and Pathology of the Gastrointestinal Tract.
Int J Mol Sci
; 24(1)2022 Dec 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-36613619
5.
The Role of Inflammatory Mediators in the Development of Gastrointestinal Motility Disorders.
Int J Mol Sci
; 23(13)2022 Jun 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-35805922
6.
Glucose-based spiro-oxathiazoles as in vivo anti-hyperglycemic agents through glycogen phosphorylase inhibition.
Org Biomol Chem
; 18(5): 931-940, 2020 02 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-31922157
7.
Synthesis of New C- and N-ß-d-Glucopyranosyl Derivatives of Imidazole, 1,2,3-Triazole and Tetrazole, and Their Evaluation as Inhibitors of Glycogen Phosphorylase.
Molecules
; 23(3)2018 Mar 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-29543771
8.
3-Glucosylated 5-amino-1,2,4-oxadiazoles: synthesis and evaluation as glycogen phosphorylase inhibitors.
Beilstein J Org Chem
; 11: 499-503, 2015.
Artículo
en Inglés
| MEDLINE | ID: mdl-25977724
9.
Glucopyranosylidene-spiro-iminothiazolidinone, a new bicyclic ring system: synthesis, derivatization, and evaluation for inhibition of glycogen phosphorylase by enzyme kinetic and crystallographic methods.
Bioorg Med Chem
; 22(15): 4028-41, 2014 Aug 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-25009003
10.
Synthesis of tartaric acid analogues of FR258900 and their evaluation as glycogen phosphorylase inhibitors.
Bioorg Med Chem Lett
; 23(6): 1789-92, 2013 Mar 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-23395662
11.
Synthesis, enzyme kinetics and computational evaluation of N-(ß-D-glucopyranosyl) oxadiazolecarboxamides as glycogen phosphorylase inhibitors.
Bioorg Med Chem
; 21(18): 5738-47, 2013 Sep 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-23938052
12.
N-(4-Substituted-benzoyl)-N'-(ß-d-glucopyranosyl)ureas as inhibitors of glycogen phosphorylase: Synthesis and evaluation by kinetic, crystallographic, and molecular modelling methods.
Bioorg Med Chem
; 20(5): 1801-16, 2012 Mar 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-22325154
13.
Dual-Target Compounds against Type 2 Diabetes Mellitus: Proof of Concept for Sodium Dependent Glucose Transporter (SGLT) and Glycogen Phosphorylase (GP) Inhibitors.
Pharmaceuticals (Basel)
; 14(4)2021 Apr 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-33920838
14.
Synthesis of 1-(D-glucopyranosyl)-1,2,3-triazoles and their evaluation as glycogen phosphorylase inhibitors.
Bioorg Med Chem
; 18(3): 1171-80, 2010 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-20080412
15.
CXCL1 is upregulated during the development of ileus resulting in decreased intestinal contractile activity.
Neurogastroenterol Motil
; 32(3): e13757, 2020 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-31722447
16.
Glycogen phosphorylase inhibitor, 2,3-bis[(2E)-3-(4-hydroxyphenyl)prop-2-enamido] butanedioic acid (BF142), improves baseline insulin secretion of MIN6 insulinoma cells.
PLoS One
; 15(9): e0236081, 2020.
Artículo
en Inglés
| MEDLINE | ID: mdl-32960890
17.
Synthesis and glycogen phosphorylase inhibitory activity of N-(beta-D-glucopyranosyl)amides possessing 1,4-benzodioxane moiety.
Bioorg Med Chem
; 17(18): 6738-41, 2009 Sep 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-19703777
18.
Synthesis and structure-activity relationships of C-glycosylated oxadiazoles as inhibitors of glycogen phosphorylase.
Bioorg Med Chem
; 17(13): 4773-85, 2009 Jul 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-19450985
19.
Glucose-based spiro-heterocycles as potent inhibitors of glycogen phosphorylase.
Bioorg Med Chem
; 17(15): 5696-707, 2009 Aug 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-19574053
20.
Synthesis of C-ß-d-glucopyranosyl derivatives of some fused azoles for the inhibition of glycogen phosphorylase.
Carbohydr Res
; 472: 33-41, 2019 Jan 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-30453096