Detalles de la búsqueda
1.
The Marine-Derived Fungus Clonostachys rosea, Source of a Rare Conjugated 4-Me-6E,8E-hexadecadienoic Acid Reducing Viability of MCF-7 Breast Cancer Cells and Gene Expression of Lipogenic Enzymes.
Mar Drugs
; 13(8): 4934-48, 2015 Aug 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-26258780
2.
Synthesis and in vitro antifungal evaluation of 2-(2,4-difluorophenyl)-1-[(1H-indol-3-ylmethyl)methylamino]-3-(1H-1,2,4-triazol-1-yl)propan-2-ols.
J Enzyme Inhib Med Chem
; 26(2): 261-9, 2011 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-20695753
3.
Synthesis of N-aryl-3-(indol-3-yl)propanamides and their immunosuppressive activities.
Bioorg Med Chem Lett
; 20(17): 5203-6, 2010 Sep 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-20655209
4.
A novel indole-3-propanamide exerts its immunosuppressive activity by inhibiting JAK3 in T cells.
J Pharmacol Exp Ther
; 331(2): 710-6, 2009 Nov.
Artículo
en Inglés
| MEDLINE | ID: mdl-19710367
5.
Indole carboxamides inhibit bovine testes hyaluronidase at pH 7.0 and indole acetamides activate the enzyme at pH 3.5 by different mechanisms.
J Enzyme Inhib Med Chem
; 23(5): 719-27, 2008 Oct.
Artículo
en Inglés
| MEDLINE | ID: mdl-18821259
6.
N-Pyridinyl(methyl)-indole-1- or 3-propanamides and propenamides acting as topical and systemic inflammation inhibitors.
J Enzyme Inhib Med Chem
; 23(5): 728-38, 2008 Oct.
Artículo
en Inglés
| MEDLINE | ID: mdl-18821260
7.
Design, synthesis and evaluation of new 6-substituted-5-benzyloxy-4-oxo-4H-pyran-2-carboxamides as potential Src inhibitors.
J Enzyme Inhib Med Chem
; 23(5): 629-40, 2008 Oct.
Artículo
en Inglés
| MEDLINE | ID: mdl-18686137
8.
Synthetic N-pyridinyl(methyl)-indol-3-ylpropanamides as new potential immunosuppressive agents.
Eur J Med Chem
; 42(5): 686-93, 2007 May.
Artículo
en Inglés
| MEDLINE | ID: mdl-17316917
9.
Novel 1,6-naphthyridin-2(1H)-ones as potential anticancer agents targeting Hsp90.
Eur J Med Chem
; 119: 17-33, 2016 Aug 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-27153346
10.
Synthesis and biological evaluation of N-aryl-7-methoxybenzo[b]furo[3,2-d]pyrimidin-4-amines and their N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amine analogues as dual inhibitors of CLK1 and DYRK1A kinases.
Eur J Med Chem
; 59: 283-95, 2013 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-23237976
11.
Discovery of a novel broad-spectrum antifungal agent derived from albaconazole.
ACS Med Chem Lett
; 4(2): 288-92, 2013 Feb 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-24900660
12.
Synthesis and biological evaluation of N-arylbenzo[b]thieno[3,2-d]pyrimidin-4-amines and their pyrido and pyrazino analogues as Ser/Thr kinase inhibitors.
Eur J Med Chem
; 58: 171-83, 2012 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-23124214
13.
Design, synthesis, and biological evaluation of 1-[(biarylmethyl)methylamino]-2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-2-ols as potent antifungal agents: new insights into structure-activity relationships.
ChemMedChem
; 6(10): 1806-15, 2011 Oct 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-21748853
14.
Design, synthesis, and in vitro antifungal activity of 1-[(4-substituted-benzyl)methylamino]-2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-2-ols.
ChemMedChem
; 6(5): 816-25, 2011 May 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-21370476
15.
Synthesis and antifungal activities of new fluconazole analogues with azaheterocycle moiety.
Bioorg Med Chem Lett
; 17(13): 3686-9, 2007 Jul 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-17482460
16.
Synthesis and biological evaluation of 5-[(aryl)(1H-imidazol-1-yl)methyl]-1H-indoles: potent and selective aromatase inhibitors.
Bioorg Med Chem Lett
; 16(5): 1134-7, 2006 Mar 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-16380254
17.
Synthesis and primary cytotoxicity evaluation of arylmethylenenaphthofuranones derivatives.
J Enzyme Inhib Med Chem
; 21(3): 313-25, 2006 Jun.
Artículo
en Inglés
| MEDLINE | ID: mdl-16918079
18.
Potential inhibitors of angiogenesis. Part II: 3-(azolylmethylene)-2,3-dihydrobenzo[b]furan-2-ones.
J Enzyme Inhib Med Chem
; 18(3): 253-7, 2003 Jun.
Artículo
en Inglés
| MEDLINE | ID: mdl-14506916
19.
New N-pyridinyl(methyl)-indolalkanamides acting as topical inflammation inhibitors.
Bioorg Med Chem Lett
; 14(21): 5441-4, 2004 Nov 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-15454241
20.
New N-pyridinyl(methyl)-N1-substituted-3-indolepropanamides acting as topical and systemic anti-inflammatory agents.
J Enzyme Inhib Med Chem
; 18(2): 201-8, 2003 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-12943205