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1.
Development of new thieno[2,3-d]pyrimidines as dual EGFR and STAT3 inhibitors endowed with anticancer and pro-apoptotic activities.
Bioorg Chem
; 143: 107101, 2024 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-38183682
2.
Novel 4-(2-arylidenehydrazineyl)thienopyrimidine derivatives as anticancer EGFR inhibitors: Design, synthesis, biological evaluation, kinome selectivity and in silico insights.
Bioorg Chem
; 140: 106799, 2023 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-37625210
3.
Discovery of novel enasidenib analogues targeting inhibition of mutant isocitrate dehydrogenase 2 as antileukaemic agents.
J Enzyme Inhib Med Chem
; 38(1): 2157411, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36629449
4.
Recruitment of hexahydroquinoline as anticancer scaffold targeting inhibition of wild and mutants EGFR (EGFRWT, EGFRT790M, and EGFRL858R).
J Enzyme Inhib Med Chem
; 38(1): 2241674, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-37548154
5.
Discovery of new symmetrical and asymmetrical nitrile-containing 1,4-dihydropyridine derivatives as dual kinases and P-glycoprotein inhibitors: synthesis, in vitro assays, and in silico studies.
J Enzyme Inhib Med Chem
; 37(1): 2489-2511, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36093880
6.
Revisiting ageless antiques; synthesis, biological evaluation, docking simulation and mechanistic insights of 1,4-Dihydropyridines as anticancer agents.
Bioorg Chem
; 114: 105054, 2021 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-34146919
7.
Design, synthesis, and molecular docking study of new monastrol analogues as kinesin spindle protein inhibitors.
Arch Pharm (Weinheim)
; 353(8): e2000060, 2020 Aug.
Artículo
en Inglés
| MEDLINE | ID: mdl-32452567
8.
Design, synthesis, and bioactivity of dihydropyrimidine derivatives as kinesin spindle protein inhibitors.
Bioorg Med Chem
; 27(23): 115126, 2019 12 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-31648875
9.
Corrigendum to "Design, synthesis, and bioactivity of dihydropyrimidine derivatives as kinesin spindle protein inhibitors" [Bioorg. Med. Chem. 27 (2019) 115126].
Bioorg Med Chem
; 28(19): 115687, 2020 Oct 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-32826133
10.
Corrigendum to "Design, synthesis, and bioactivity of dihydropyrimidine derivatives as kinesin spindle protein inhibitors" [Bioorg. Med. Chem. 27 (2019) 115126].
Bioorg Med Chem
; 28(2): 115255, 2020 Jan 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-31862309
11.
A new framework for novel analogues of pazopanib as potent and selective human carbonic anhydrase inhibitors: Design, repurposing rational, synthesis, crystallographic, in vivo and in vitro biological assessments.
Eur J Med Chem
; 274: 116527, 2024 Aug 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-38810335
12.
Discovery and Mechanistic Studies of Dual-Target Hits for Carbonic Anhydrase IX and VEGFR-2 as Potential Agents for Solid Tumors: X-ray, In Vitro, In Vivo, and In Silico Investigations of Coumarin-Based Thiazoles.
J Med Chem
; 67(9): 7406-7430, 2024 May 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-38642371
13.
Synthesis and anticancer activity of new benzensulfonamides incorporating s-triazines as cyclic linkers for inhibition of carbonic anhydrase IX.
Sci Rep
; 12(1): 16756, 2022 10 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-36202955
14.
Structurally Diverse Histone Deacetylase Photoreactive Probes: Design, Synthesis, and Photolabeling Studies in Live Cells and Tissue.
ChemMedChem
; 14(11): 1096-1107, 2019 06 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-30921497
15.
Determination of calcium oxalate (mono- and dihydrate) in mixtures with magnesium ammonium phosphate or uric acid: the use of simultaneous thermal analysis in urinary calculi.
Clin Chim Acta
; 334(1-2): 117-29, 2003 Aug.
Artículo
en Inglés
| MEDLINE | ID: mdl-12867282
16.
Synthesis and dopamine transporter binding of 2beta-isopropyl ester analogs of cocaine.
Eur J Med Chem
; 37(2): 171-6, 2002 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-11858849
17.
Fluorescence Spectrometric Determination of Drugs Containing α-Methylene Sulfone/Sulfonamide Functional Groups Using N-Methylnicotinamide Chloride as a Fluorogenic Agent.
Int J Anal Chem
; 2011: 840178, 2011.
Artículo
en Inglés
| MEDLINE | ID: mdl-21647288
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