Detalles de la búsqueda
1.
Essential Oils from Mediterranean Plants Inhibit In Vitro Monocyte Adhesion to Endothelial Cells from Umbilical Cords of Females with Gestational Diabetes Mellitus.
Int J Mol Sci
; 24(8)2023 Apr 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-37108387
2.
Molecular Docking Assessment of Cathinones as 5-HT2AR Ligands: Developing of Predictive Structure-Based Bioactive Conformations and Three-Dimensional Structure-Activity Relationships Models for Future Recognition of Abuse Drugs.
Molecules
; 28(17)2023 Aug 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-37687065
3.
Bovine Serum Amine Oxidase and Polyamine Analogues: Chemical Synthesis and Biological Evaluation Integrated with Molecular Docking and 3-D QSAR Studies.
J Chem Inf Model
; 62(16): 3910-3927, 2022 08 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-35948439
4.
Heterocycle-containing tranylcypromine derivatives endowed with high anti-LSD1 activity.
J Enzyme Inhib Med Chem
; 37(1): 973-985, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-35317680
5.
Current HDAC Inhibitors in Clinical Trials.
Chimia (Aarau)
; 76(5): 448-453, 2022 May 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-38069716
6.
Properly Substituted Cyclic Bis-(2-bromobenzylidene) Compounds Behaved as Dual p300/CARM1 Inhibitors and Induced Apoptosis in Cancer Cells.
Molecules
; 25(14)2020 Jul 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-32650558
7.
Six Years (2012-2018) of Researches on Catalytic EZH2 Inhibitors: The Boom of the 2-Pyridone Compounds.
Chem Rec
; 18(12): 1818-1832, 2018 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-30338896
8.
N-((1,3-Diphenyl-1H-pyrazol-4-yl)methyl)anilines: A novel class of anti-RSV agents.
Bioorg Med Chem Lett
; 25(11): 2401-4, 2015 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-25913116
9.
Selenium-containing compounds: a new hope for innovative treatments in Alzheimer's disease and Parkinson's disease.
Drug Discov Today
; : 104062, 2024 Jun 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-38871111
10.
Uracil- and Pyridine-Containing HDAC Inhibitors Displayed Cytotoxicity in Colorectal and Glioblastoma Cancer Stem Cells.
ChemMedChem
; : e202300655, 2024 Mar 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-38529661
11.
Theileria parasites sequester host eIF5A to escape elimination by host-mediated autophagy.
Nat Commun
; 15(1): 2235, 2024 Mar 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-38472173
12.
Correction: Zwergel et al. Novel Quinoline Compounds Active in Cancer Cells through Coupled DNA Methyltransferase Inhibition and Degradation. Cancers 2020, 12, 447.
Cancers (Basel)
; 16(6)2024 Mar 21.
Artículo
en Inglés
| MEDLINE | ID: mdl-38539577
13.
First-in-Class Selenium-Containing Potent Serotonin Receptor 5-HT6 Agents with a Beneficial Neuroprotective Profile against Alzheimer's Disease.
J Med Chem
; 67(2): 1580-1610, 2024 Jan 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-38190615
14.
Design, synthesis, and in vitro hMAO-B inhibitory evaluation of some 1-methyl-3,5-diphenyl-4,5-dihydro-1H-pyrazoles.
Bioorg Med Chem Lett
; 23(18): 5128-30, 2013 Sep 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-23927971
15.
PD-L1 small-molecule modulators: A new hope in epigenetic-based multidrug cancer therapy?
Drug Discov Today
; 28(2): 103435, 2023 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-36370994
16.
LSD1 inhibitors for cancer treatment: Focus on multi-target agents and compounds in clinical trials.
Front Pharmacol
; 14: 1120911, 2023.
Artículo
en Inglés
| MEDLINE | ID: mdl-36817147
17.
Histone deacetylase 10: A polyamine deacetylase from the crystal structure to the first inhibitors.
Curr Opin Struct Biol
; 82: 102668, 2023 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-37542907
18.
Screening of the activity of sixty essential oils against plasmodium early mosquito stages in vitro and machine learning analysis reveals new putative inhibitors of malaria parasites.
Int J Parasitol Drugs Drug Resist
; 23: 87-93, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-38000094
19.
Chemically Diverse S. mansoni HDAC8 Inhibitors Reduce Viability in Worm Larval and Adult Stages.
ChemMedChem
; 18(3): e202200510, 2023 02 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-36250286
20.
Novel 1,4-Dihydropyridines as Specific Binders and Activators of SIRT3 Impair Cell Viability and Clonogenicity and Downregulate Hypoxia-Induced Targets in Cancer Cells.
J Med Chem
; 66(14): 9622-9641, 2023 07 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-37439550