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1.
Discovery of Small Molecule Drugs Targeting the Biogenesis of microRNA-155 for the Treatment of Systemic Lupus Erythematosus.
Chimia (Aarau)
; 74(10): 798-802, 2020 Oct 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-33115563
2.
Evolution of novel tricyclic CRTh2 receptor antagonists from a (E)-2-cyano-3-(1H-indol-3-yl)acrylamide scaffold.
Bioorg Med Chem Lett
; 23(4): 944-8, 2013 Feb 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-23324405
3.
Novel 2-(2-(benzylthio)-1H-benzo[d]imidazol-1-yl)acetic acids: discovery and hit-to-lead evolution of a selective CRTh2 receptor antagonist chemotype.
Bioorg Med Chem Lett
; 22(14): 4660-4, 2012 Jul 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-22726929
4.
Protein kinases as targets for anticancer agents: from inhibitors to useful drugs.
Pharmacol Ther
; 93(2-3): 79-98, 2002.
Artículo
en Inglés
| MEDLINE | ID: mdl-12191602
5.
Verification of the Major Metabolic Oxidation Path for the Naphthoyl Group in Chemoattractant Receptor-Homologous Molecule Expressed on Th2 Cells (CRTh2) Antagonist 2-(2-(1-Naphthoyl)-8-fluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5(2H)-yl)acetic Acid (Setipiprant/ACT-129968).
J Med Chem
; 58(20): 8011-35, 2015 Oct 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-26398218
6.
Structure-based design and synthesis of 2-benzylidene-benzofuran-3-ones as flavopiridol mimics.
J Med Chem
; 45(9): 1741-7, 2002 Apr 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-11960485
7.
Identification of 2-(2-(1-naphthoyl)-8-fluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5(2H)-yl)acetic acid (setipiprant/ACT-129968), a potent, selective, and orally bioavailable chemoattractant receptor-homologous molecule expressed on Th2 cells (CRTH2) antagonist.
J Med Chem
; 56(12): 4899-911, 2013 Jun 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-23721423
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