Detalles de la búsqueda
1.
Quinazolinone-based benzenesulfonamides with low toxicity and high affinity as monoamine oxidase-A inhibitors: Synthesis, biological evaluation and induced-fit docking studies.
Bioorg Chem
; 124: 105822, 2022 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-35500503
2.
Investigation of carbonic anhydrase inhibitory effects and cytotoxicities of pyrazole-based hybrids carrying hydrazone and zinc-binding benzenesulfonamide pharmacophores.
Bioorg Chem
; 127: 105969, 2022 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-35926240
3.
Synthesis and in vitro carbonic anhydrases and acetylcholinesterase inhibitory activities of novel imidazolinone-based benzenesulfonamides.
Arch Pharm (Weinheim)
; 354(4): e2000375, 2021 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-33283898
4.
Synthesis of benzamide derivatives with thiourea-substituted benzenesulfonamides as carbonic anhydrase inhibitors.
Arch Pharm (Weinheim)
; 354(2): e2000230, 2021 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-33043495
5.
Monoamine Oxidase (MAO) as a Potential Target for Anticancer Drug Design and Development.
Molecules
; 26(19)2021 Oct 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-34641563
6.
Synthesis, structure elucidation, and in vitro pharmacological evaluation of novel polyfluoro substituted pyrazoline type sulfonamides as multi-target agents for inhibition of acetylcholinesterase and carbonic anhydrase I and II enzymes.
Bioorg Chem
; 96: 103627, 2020 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-32058104
7.
Novel sulphonamides incorporating triazene moieties show powerful carbonic anhydrase I and II inhibitory properties.
J Enzyme Inhib Med Chem
; 35(1): 325-329, 2020 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-31813300
8.
Deciphering binding mechanism between bovine serum albumin and new pyrazoline compound K4.
Luminescence
; 35(4): 534-541, 2020 Jun.
Artículo
en Inglés
| MEDLINE | ID: mdl-31883290
9.
Investigation of inhibitory properties of some hydrazone compounds on hCA I, hCA II and AChE enzymes.
Bioorg Chem
; 86: 316-321, 2019 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-30743172
10.
Synthesis, biological evaluation and in silico modelling studies of 1,3,5-trisubstituted pyrazoles carrying benzenesulfonamide as potential anticancer agents and selective cancer-associated hCA IX isoenzyme inhibitors.
Bioorg Chem
; 92: 103222, 2019 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-31499260
11.
Synthesis and biological evaluation of some new mono Mannich bases with piperazines as possible anticancer agents and carbonic anhydrase inhibitors.
Bioorg Chem
; 90: 103095, 2019 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-31288135
12.
Synthesis and bioactivities of pyrazoline benzensulfonamides as carbonic anhydrase and acetylcholinesterase inhibitors with low cytotoxicity.
Bioorg Chem
; 84: 511-517, 2019 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-30605787
13.
New phenolic Mannich bases with piperazines and their bioactivities.
Bioorg Chem
; 90: 103057, 2019 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-31226471
14.
Synthesis, cytotoxicities, and carbonic anhydrase inhibition potential of 6-(3-aryl-2-propenoyl)-2(3H)-benzoxazolones.
J Enzyme Inhib Med Chem
; 34(1): 1722-1729, 2019 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-31576761
15.
Anticancer effects of new dibenzenesulfonamides by inducing apoptosis and autophagy pathways and their carbonic anhydrase inhibitory effects on hCA I, hCA II, hCA IX, hCA XII isoenzymes.
Bioorg Chem
; 78: 290-297, 2018 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-29621641
16.
Curcumin analogue 1,5-bis(4-hydroxy-3-((4-methylpiperazin-1-yl)methyl)phenyl)penta-1,4-dien-3-one mediates growth arrest and apoptosis by targeting the PI3K/AKT/mTOR and PKC-theta signaling pathways in human breast carcinoma cells.
Bioorg Chem
; 78: 46-57, 2018 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-29533214
17.
New anticancer drug candidates sulfonamides as selective hCA IX or hCA XII inhibitors.
Bioorg Chem
; 77: 411-419, 2018 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-29427856
18.
Synthesis, carbonic anhydrase I and II inhibition studies of the 1,3,5-trisubstituted-pyrazolines.
J Enzyme Inhib Med Chem
; 32(1): 189-192, 2017 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-27774818
19.
Microwave-assisted synthesis and bioevaluation of new sulfonamides.
J Enzyme Inhib Med Chem
; 32(1): 369-374, 2017 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-28260401
20.
Designing, synthesis and bioactivities of 4-[3-(4-hydroxyphenyl)-5-aryl-4,5-dihydro-pyrazol-1-yl]benzenesulfonamides.
J Enzyme Inhib Med Chem
; 32(1): 169-175, 2017 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-27774817