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1.
Discovery and Optimization of Pyridazinones as PI3Kδ Selective Inhibitors for Administration by Inhalation.
J Med Chem
; 2024 Jun 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-38907711
2.
Functionalized pyrazoles and pyrazolo[3,4-d]pyridazinones: Synthesis and evaluation of their phosphodiesterase 4 inhibitory activity.
Bioorg Med Chem
; 18(10): 3506-17, 2010 May 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-20413313
3.
Atropisomerism and Conformational Equilibria: Impact on PI3Kδ Inhibition of 2-((6-Amino-9H-purin-9-yl)methyl)-5-methyl-3-(o-tolyl)quinazolin-4(3H)-one (IC87114) and Its Conformationally Restricted Analogs.
J Med Chem
; 60(10): 4304-4315, 2017 05 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-28489362
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