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1.
Discovery of a septin-4 covalent binder with antimetastatic activity in a mouse model of melanoma.
Bioorg Chem
; 144: 107164, 2024 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-38306824
2.
Investigation into the Use of Encorafenib to Develop Potential PROTACs Directed against BRAFV600E Protein.
Molecules
; 27(23)2022 Dec 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-36500607
3.
Chemical Modulation of the 1-(Piperidin-4-yl)-1,3-dihydro-2H-benzo[d]imidazole-2-one Scaffold as a Novel NLRP3 Inhibitor.
Molecules
; 26(13)2021 Jun 29.
Artículo
en Inglés
| MEDLINE | ID: mdl-34209843
4.
Development of covalent NLRP3 inflammasome inhibitors: Chemistry and biological activity.
Arch Biochem Biophys
; 670: 116-139, 2019 07 30.
Artículo
en Inglés
| MEDLINE | ID: mdl-30448387
5.
Discovery of a novel 1,3,4-oxadiazol-2-one-based NLRP3 inhibitor as a pharmacological agent to mitigate cardiac and metabolic complications in an experimental model of diet-induced metaflammation.
Eur J Med Chem
; 257: 115542, 2023 Sep 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-37290185
6.
A Comparative Study on the Efficacy of NLRP3 Inflammasome Signaling Inhibitors in a Pre-clinical Model of Bowel Inflammation.
Front Pharmacol
; 9: 1405, 2018.
Artículo
en Inglés
| MEDLINE | ID: mdl-30559669
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