Detalles de la búsqueda
1.
Boron-containing carbonic anhydrases inhibitors.
Bioorg Chem
; 143: 106976, 2024 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-38000350
2.
Identification of thienopyrimidine derivatives tethered with sulfonamide and other moieties as carbonic anhydrase inhibitors: Design, synthesis and anti-proliferative activity.
Bioorg Chem
; 144: 107089, 2024 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-38237393
3.
Cloning, expression, and purification of an α-carbonic anhydrase from Toxoplasma gondii to unveil its kinetic parameters and anion inhibition profile.
J Enzyme Inhib Med Chem
; 39(1): 2346523, 2024 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-38847581
4.
In-vitro and in-silico investigations of SLC-0111 hydrazinyl analogs as human carbonic anhydrase I, II, IX, and XII inhibitors.
Arch Pharm (Weinheim)
; : e2400157, 2024 May 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-38713910
5.
1,2,3-Triazole-based esters and carboxylic acids as nonclassical carbonic anhydrase inhibitors capable of cathepsin B inhibition.
Arch Pharm (Weinheim)
; 357(3): e2300372, 2024 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-38012535
6.
Potent and selective carbonic anhydrase inhibition activities of pyrazolones bearing benzenesulfonamides.
Bioorg Med Chem Lett
; 95: 129479, 2023 10 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-37704010
7.
Design and synthesis of sulfonamides incorporating a biotin moiety: Carbonic anhydrase inhibitory effects, antiproliferative activity and molecular modeling studies.
Bioorg Med Chem
; 94: 117467, 2023 Oct 30.
Artículo
en Inglés
| MEDLINE | ID: mdl-37722299
8.
Discovery of the first-in-class potent and isoform-selective human carbonic anhydrase III inhibitors.
J Enzyme Inhib Med Chem
; 38(1): 2202360, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-37092262
9.
Inhibition studies with simple and complex (in)organic anions of the γ-carbonic anhydrase from Mammaliicoccus (Staphylococcus) sciuri, MscCAγ.
J Enzyme Inhib Med Chem
; 38(1): 2173748, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36719031
10.
Inhibition of pathogenic bacterial carbonic anhydrases by monothiocarbamates.
J Enzyme Inhib Med Chem
; 38(1): 2284119, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-37994421
11.
Potent inhibitors of tumor associated carbonic anhydrases endowed with cathepsin B inhibition.
Arch Pharm (Weinheim)
; 356(11): e2300349, 2023 Nov.
Artículo
en Inglés
| MEDLINE | ID: mdl-37704930
12.
Conformationally Restricted Glycoconjugates Derived from Arylsulfonamides and Coumarins: New Families of Tumour-Associated Carbonic Anhydrase Inhibitors.
Int J Mol Sci
; 24(11)2023 May 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-37298353
13.
4-(3-Alkyl/benzyl-guanidino)benzenesulfonamides as selective carbonic anhydrase VII inhibitors.
J Enzyme Inhib Med Chem
; 37(1): 1568-1576, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-35635139
14.
Coumarins inhibit η-class carbonic anhydrase from Plasmodium falciparum.
J Enzyme Inhib Med Chem
; 37(1): 680-685, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-35139744
15.
Coumarins effectively inhibit bacterial α-carbonic anhydrases.
J Enzyme Inhib Med Chem
; 37(1): 333-338, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-34979838
16.
Inhibition studies of bacterial α-carbonic anhydrases with phenols.
J Enzyme Inhib Med Chem
; 37(1): 666-671, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-35139743
17.
Dithiocarbamates effectively inhibit the α-carbonic anhydrase from Neisseria gonorrhoeae.
J Enzyme Inhib Med Chem
; 37(1): 1-8, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-34894954
18.
May Sulfonamide Inhibitors of Carbonic Anhydrases from Mammaliicoccus sciuri Prevent Antimicrobial Resistance Due to Gene Transfer to Other Harmful Staphylococci?
Int J Mol Sci
; 23(22)2022 Nov 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-36430304
19.
Continued Structural Exploration of Sulfocoumarin as Selective Inhibitor of Tumor-Associated Human Carbonic Anhydrases IX and XII.
Molecules
; 27(13)2022 Jun 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-35807318
20.
Aromatic Sulfonamides including a Sulfonic Acid Tail: New Membrane Impermeant Carbonic Anhydrase Inhibitors for Targeting Selectively the Cancer-Associated Isoforms.
Int J Mol Sci
; 23(1)2021 Dec 31.
Artículo
en Inglés
| MEDLINE | ID: mdl-35008884