Detalles de la búsqueda
1.
Cloning and functional analysis of a polymorphic variant of the ovine Mel 1a melatonin receptor.
Biochim Biophys Acta
; 1356(3): 299-307, 1997 May 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-9194573
2.
[Melatoninergic receptor agonists and antagonists: pharmacological aspects and therapeutic perspective]. / Agonistes et antagonistes des récepteurs mélatoninergiques: effets pharmacologiques et perspectives thérapeutiques.
Ann Pharm Fr
; 63(6): 385-400, 2005 Nov.
Artículo
en Francés
| MEDLINE | ID: mdl-16292232
3.
Toxicology of melatonin.
J Biol Rhythms
; 12(6): 697-706, 1997 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-9406047
4.
Effects of a novel melatonin analog on circadian rhythms of body temperature and activity in young, middle-aged, and old rats.
Neurobiol Aging
; 14(6): 565-9, 1993.
Artículo
en Inglés
| MEDLINE | ID: mdl-8295659
5.
Identification of Mel1a melatonin receptors in the human embryonic kidney cell line HEK293: evidence of G protein-coupled melatonin receptors which do not mediate the inhibition of stimulated cyclic AMP levels.
FEBS Lett
; 407(1): 121-6, 1997 Apr 21.
Artículo
en Inglés
| MEDLINE | ID: mdl-9141494
6.
3,4-Dihydro-3-amino-2H-1-benzopyran derivatives as 5-HT1A receptor ligands and potential anxiolytic agents. 1. Synthesis and structure--activity relationship studies.
J Med Chem
; 37(12): 1779-93, 1994 Jun 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-7912735
7.
Novel and selective partial agonists of 5-HT3 receptors. 2. Synthesis and biological evaluation of piperazinopyridopyrrolopyrazines, piperazinopyrroloquinoxalines, and piperazinopyridopyrroloquinoxalines.
J Med Chem
; 40(12): 1808-19, 1997 Jun 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-9191957
8.
Novel benzothiazolin-2-one and benzoxazin-3-one arylpiperazine derivatives with mixed 5HT1A/D2 affinity as potential atypical antipsychotics.
J Med Chem
; 41(12): 2010-8, 1998 Jun 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-9622542
9.
Novel selective and partial agonists of 5-HT3 receptors. Part 1. Synthesis and biological evaluation of piperazinopyrrolothienopyrazines.
J Med Chem
; 39(10): 2068-80, 1996 May 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-8642566
10.
Novel indole-2-carboxamide and cycloalkeno[1,2-b]indole derivatives. Structure-activity relationships for high inhibition of human LDL peroxidation.
J Med Chem
; 40(8): 1201-10, 1997 Apr 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-9111294
11.
3-amino-3,4-dihydro-2H-1-benzopyran derivatives as 5-HT1A receptor ligands and potential anxiolytic agents. 2. Synthesis and quantitative structure-activity relationship studies of spiro[pyrrolidine- and piperidine-2,3'(2'H)-benzopyrans].
J Med Chem
; 39(21): 4285-98, 1996 Oct 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-8863806
12.
Design and synthesis of imidazoline derivatives active on glucose homeostasis in a rat model of type II diabetes. 1. Synthesis and biological activities of N-benzyl-N'-(arylalkyl)-2-(4',5'-dihydro-1'H-imidazol-2'-yl)piperazines .
J Med Chem
; 40(23): 3793-803, 1997 Nov 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-9371245
13.
Design and synthesis of imidazoline derivatives active on glucose homeostasis in a rat model of type II diabetes. 2. Syntheses and biological activities of 1,4-dialkyl-, 1,4-dibenzyl, and 1-benzyl-4-alkyl-2-(4',5'-dihydro-1'H-imidazol-2'-yl)piperazines and isosteric analogues of imidazoline.
J Med Chem
; 42(9): 1587-603, 1999 May 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-10229628
14.
Stimulation of insulin release from the MIN6 cell line by a new imidazoline compound, S-21663: evidence for the existence of a novel imidazoline site in beta cells.
Br J Pharmacol
; 122(4): 786-91, 1997 Oct.
Artículo
en Inglés
| MEDLINE | ID: mdl-9375978
15.
Studies on the vasoconstrictor action of melatonin and putative melatonin receptor ligands in the tail artery of juvenile Wistar rats.
Br J Pharmacol
; 122(7): 1299-306, 1997 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-9421275
16.
In vitro mechanism of action on insulin release of S-22068, a new putative antidiabetic compound.
Br J Pharmacol
; 128(5): 1021-6, 1999 Nov.
Artículo
en Inglés
| MEDLINE | ID: mdl-10556939
17.
Potent antihyperglycaemic property of a new imidazoline derivative S-22068 (PMS 847) in a rat model of NIDDM.
Br J Pharmacol
; 124(8): 1591-6, 1998 Aug.
Artículo
en Inglés
| MEDLINE | ID: mdl-9756373
18.
Anticonflict and discriminative stimulus effects in the pigeon of a new methoxy-chroman 5-HT1A agonist, (+)S 20244 and its enantiomers (+)S 20499 and (-)S 20500.
Psychopharmacology (Berl)
; 116(1): 73-8, 1994 Sep.
Artículo
en Inglés
| MEDLINE | ID: mdl-7862933
19.
Dose dependent effects of S-20098, a melatonin agonist, on direction of re-entrainment of rat circadian activity rhythms.
Psychopharmacology (Berl)
; 118(4): 385-90, 1995 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-7568624
20.
Melatonin receptors mediate contraction of a rat cerebral artery.
Neuroreport
; 8(18): 3847-9, 1997 Dec 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-9462453