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1.
A novel N-heterocycles substituted oseltamivir derivatives as potent inhibitors of influenza virus neuraminidase: discovery, synthesis and biological evaluation.
J Enzyme Inhib Med Chem
; 38(1): 2277135, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-37955306
2.
Discovery of Novel Boron-Containing N-Substituted Oseltamivir Derivatives as Anti-Influenza A Virus Agents for Overcoming N1-H274Y Oseltamivir-Resistant.
Molecules
; 27(19)2022 Sep 29.
Artículo
en Inglés
| MEDLINE | ID: mdl-36234966
3.
Iterative Optimization and Structure-Activity Relationship Studies of Oseltamivir Amino Derivatives as Potent and Selective Neuraminidase Inhibitors via Targeting 150-Cavity.
J Med Chem
; 65(17): 11550-11573, 2022 09 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-35939763
4.
Identification of C5-NH2 Modified Oseltamivir Derivatives as Novel Influenza Neuraminidase Inhibitors with Highly Improved Antiviral Activities and Favorable Druggability.
J Med Chem
; 64(24): 17992-18009, 2021 12 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-34735766
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