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1.
Exploring the Antiproliferative Potency of Pyrido[2,3-d]Pyrimidine Derivatives: Studies on Design, Synthesis, Anticancer Evaluation, SAR, Docking, and DFT Calculations.
Chem Biodivers
; 21(2): e202301682, 2024 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-38084395
2.
Synthesis and Antimicrobial, Anticancer and Anti-Oxidant Activities of Novel 2,3-Dihydropyrido[2,3-d]pyrimidine-4-one and Pyrrolo[2,1-b][1,3]benzothiazole Derivatives via Microwave-Assisted Synthesis.
Molecules
; 27(4)2022 Feb 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-35209034
3.
Novel pyrazole derivatives with oxa/thiadiazolyl, pyrazolyl moieties and pyrazolo[4,3-d]-pyrimidine derivatives as potential antimicrobial and anticancer agents.
Bioorg Med Chem Lett
; 26(10): 2428-2433, 2016 05 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-27080187
4.
Synthesis and Biological Evaluation of N- Pyrazolyl Derivatives and Pyrazolopyrimidine Bearing a Biologically Active Sulfonamide Moiety as Potential Antimicrobial Agent.
Molecules
; 21(9)2016 Aug 31.
Artículo
en Inglés
| MEDLINE | ID: mdl-27589717
5.
Synthesis of Novel Pyridine Bearing Biologically Active Imidiazolyl, Pyrazolyl, Oxa/thiadiazolyl and Urea Derivatives as Promising Anticancer Agents.
Curr Org Synth
; 17(1): 55-64, 2020.
Artículo
en Inglés
| MEDLINE | ID: mdl-32103718
6.
Synthesis and antitumor activity of substituted triazolo[4,3-a]pyrimidin-6-sulfonamide with an incorporated thiazolidinone moiety.
Bioorg Med Chem Lett
; 19(15): 4143-7, 2009 Aug 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-19540114
7.
Synthesis of 4-substituted pyrido[2,3-d]pyrimidin-4(1H)-one as analgesic and anti-inflammatory agents.
Bioorg Med Chem Lett
; 19(13): 3392-7, 2009 Jul 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-19481936
8.
Synthesis and evaluation of analgesic, anti-inflammatory and ulcerogenic activities of some triazolo- and 2-pyrazolyl-pyrido[2,3-d]-pyrimidines.
Acta Pharm
; 58(4): 359-78, 2008 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-19103572
9.
Synthesis and biological evaluation of thieno[2,3-d]pyrimidine derivatives for anti-inflammatory, analgesic and ulcerogenic activity.
Acta Pharm
; 57(4): 395-411, 2007 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-18165185
10.
Synthesis and evaluation of antitumor activity of new 4-substituted thieno[3,2-d]pyrimidine and thienotriazolopyrimidine derivatives.
Acta Pharm
; 67(4): 527-542, 2017 Dec 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-29337675
11.
Synthesis of thiophene and N-substituted thieno[3,2-d] pyrimidine derivatives as potent antitumor and antibacterial agents.
Acta Pharm
; 67(3): 275-292, 2017 Sep 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-28858838
12.
Simple approach to thieno[3,2-d]pyrimidines as new scaffolds of antimicrobial activities.
Acta Pharm
; 66(3): 331-51, 2016 Sep 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-27383884
13.
Synthesis of pyranopyrazolo N-glycoside and pyrazolopyranopyrimidine C-glycoside derivatives as promising antitumor and antimicrobial agents.
Acta Pharm
; 65(3): 215-33, 2015 Sep.
Artículo
en Inglés
| MEDLINE | ID: mdl-26431102
14.
Facile heterocyclic synthesis and antimicrobial activity of polysubstituted and condensed pyrazolopyranopyrimidine and pyrazolopyranotriazine derivatives.
Acta Pharm
; 65(4): 399-412, 2015 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-26677897
15.
Synthesis, in vitro antimicrobial and in vivo antitumor evaluation of novel pyrimidoquinolines and its nucleoside derivatives.
Eur J Med Chem
; 46(1): 21-30, 2011 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-21074295
16.
Synthesis of substituted thieno[2,3-d]pyrimidine-2,4-dithiones and their S-glycoside analogues as potential antiviral and antibacterial agents.
Eur J Med Chem
; 45(9): 4026-34, 2010 Sep.
Artículo
en Inglés
| MEDLINE | ID: mdl-20691339
17.
Synthesis, biological and medicinal significance of S-glycosido-thieno[2,3-d]-pyrimidines as new anti-inflammatory and analgesic agents.
Eur J Med Chem
; 45(4): 1485-93, 2010 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-20116903
18.
S- and C-nucleosidoquinazoline as new nucleoside analogs with potential analgesic and anti-inflammatory activity.
Eur J Med Chem
; 44(10): 4249-58, 2009 Oct.
Artículo
en Inglés
| MEDLINE | ID: mdl-19541393
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