Detalles de la búsqueda
1.
Effects of a dietary intervention with Mediterranean vs lacto-ovo vegetarian diets on HDL function: Results from the CARDIVEG study.
Nutr Metab Cardiovasc Dis
; 33(3): 651-658, 2023 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-36642608
2.
A New ABCB1 Inhibitor Enhances the Anticancer Effect of Doxorubicin in Both In Vitro and In Vivo Models of NSCLC.
Int J Mol Sci
; 24(2)2023 Jan 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-36674503
3.
4-Thiazolidinone Derivatives as MMP Inhibitors in Tissue Damage: Synthesis, Biological Evaluation and Docking Studies.
Molecules
; 23(2)2018 Feb 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-29443898
4.
Exploiting Free-Energy Minima to Design Novel EphA2 Protein-Protein Antagonists: From Simulation to Experiment and Return.
Chemistry
; 22(24): 8048-52, 2016 Jun 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-27139720
5.
2-Benzisothiazolylimino-5-benzylidene-4-thiazolidinones as protective agents against cartilage destruction.
Bioorg Med Chem
; 23(7): 1551-6, 2015 Apr 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-25725607
6.
Comparative Analysis of Virtual Screening Approaches in the Search for Novel EphA2 Receptor Antagonists.
Molecules
; 20(9): 17132-51, 2015 Sep 17.
Artículo
en Inglés
| MEDLINE | ID: mdl-26393553
7.
Combining ligand- and structure-based approaches for the discovery of new inhibitors of the EPHA2-ephrin-A1 interaction.
J Chem Inf Model
; 54(10): 2621-6, 2014 Oct 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-25289483
8.
Design synthesis and antibacterial activity studies of new thiadiazoloquinolone compounds.
J Enzyme Inhib Med Chem
; 29(6): 777-85, 2014 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-24506209
9.
Synthesis and structure-activity relationships of amino acid conjugates of cholanic acid as antagonists of the EphA2 receptor.
Molecules
; 18(10): 13043-60, 2013 Oct 21.
Artículo
en Inglés
| MEDLINE | ID: mdl-24152675
10.
Nucleoside Derivatives of 2,6-Diaminopurine Antivirals: Base-Modified Nucleosides with Broad-Spectrum Antimicrobial Properties.
ChemMedChem
; 18(16): e202300200, 2023 08 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-37221137
11.
Probing the effects of MR120 in preclinical chronic colitis: A first-in-class anti-IBD agent targeting the CCL20/CCR6 axis.
Eur J Pharmacol
; 945: 175613, 2023 Apr 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-36841282
12.
Synthesis and biological evaluation of tetracyclic thienopyridones as antibacterial and antitumor agents.
Bioorg Med Chem
; 19(8): 2541-8, 2011 Apr 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-21458275
13.
Heteroarylimino-4-thiazolidinones as inhibitors of cartilage degradation.
Bioorg Chem
; 39(1): 48-52, 2011 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-21208635
14.
Probucol treatment is associated with an ABCA1-independent mechanism of cholesterol efflux to lipid poor apolipoproteins from foam cell macrophages.
BBA Adv
; 1: 100003, 2021.
Artículo
en Inglés
| MEDLINE | ID: mdl-37082009
15.
Metabolic Soft Spot and Pharmacokinetics: Functionalization of C-3 Position of an Eph-Ephrin Antagonist Featuring a Bile Acid Core as an Effective Strategy to Obtain Oral Bioavailability in Mice.
Pharmaceuticals (Basel)
; 15(1)2021 Dec 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-35056098
16.
Bithiazole Inhibitors of Phosphatidylinositol 4-Kinase (PI4KIIIß) as Broad-Spectrum Antivirals Blocking the Replication of SARS-CoV-2, Zika Virus, and Human Rhinoviruses.
ChemMedChem
; 16(23): 3548-3552, 2021 12 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-34382337
17.
On the use of 2,5-dimethyl-pyrrol-1-yl-benzoic acid derivatives as EPH-ephrin antagonists.
J Virol
; 88(20): 12173, 2014 Oct.
Artículo
en Inglés
| MEDLINE | ID: mdl-25246598
18.
Synthesis and biological evaluation of tetracyclic fluoroquinolones as antibacterial and anticancer agents.
Bioorg Med Chem
; 18(16): 5873-84, 2010 Aug 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-20667744
19.
Evaluation of the Anti-Tumor Activity of Small Molecules Targeting Eph/Ephrins in APC min/J Mice.
Pharmaceuticals (Basel)
; 13(4)2020 Apr 16.
Artículo
en Inglés
| MEDLINE | ID: mdl-32316101
20.
Optimization of EphA2 antagonists based on a lithocholic acid core led to the identification of UniPR505, a new 3α-carbamoyloxy derivative with antiangiogenetic properties.
Eur J Med Chem
; 189: 112083, 2020 Mar 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-32000051