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1.
Selective antiproliferative effect of C-2 halogenated 13α-estrones on cells expressing Organic anion-transporting polypeptide 2B1 (OATP2B1).
Toxicol Appl Pharmacol
; 429: 115704, 2021 10 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-34474082
2.
Design, synthesis and biological evaluation of novel estrone phosphonates as high affinity organic anion-transporting polypeptide 2B1 (OATP2B1) inhibitors.
Bioorg Chem
; 112: 104914, 2021 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-33932771
3.
Synthesis and evaluation of AKR1C inhibitory properties of A-ring halogenated oestrone derivatives.
J Enzyme Inhib Med Chem
; 36(1): 1500-1508, 2021 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-34227437
4.
Microwave-assisted Phospha-Michael addition reactions in the 13α-oestrone series and in vitro antiproliferative properties.
J Enzyme Inhib Med Chem
; 36(1): 1931-1937, 2021 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-34445919
5.
Synthesis and evaluation of anticancer activities of 2- or 4-substituted 3-(N-benzyltriazolylmethyl)-13α-oestrone derivatives.
J Enzyme Inhib Med Chem
; 36(1): 58-67, 2021 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-33121276
6.
Synthesis, Biological Evaluation and Docking Studies of 13-Epimeric 10-fluoro- and 10-Chloroestra-1,4-dien-3-ones as Potential Aromatase Inhibitors.
Molecules
; 24(9)2019 May 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-31072017
7.
Synthesis and structure-activity relationships of 2- and/or 4-halogenated 13ß- and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis.
J Enzyme Inhib Med Chem
; 33(1): 1271-1282, 2018 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-30230387
8.
Pd-Catalyzed microwave-assisted synthesis of phosphonated 13α-estrones as potential OATP2B1, 17ß-HSD1 and/or STS inhibitors.
Beilstein J Org Chem
; 14: 2838-2845, 2018.
Artículo
en Inglés
| MEDLINE | ID: mdl-30498534
9.
Synthesis of novel 13α-estrone derivatives by Sonogashira coupling as potential 17ß-HSD1 inhibitors.
Beilstein J Org Chem
; 13: 1303-1309, 2017.
Artículo
en Inglés
| MEDLINE | ID: mdl-28694873
10.
Cytotoxic effect of 13α-estrane derivatives on breast, endometrial and ovarian cancer cell lines.
J Steroid Biochem Mol Biol
; 232: 106350, 2023 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-37315869
11.
Novel preparation of substituted oxazolines condensed to d-ring of estrane skeleton and characterization of their antiproliferative properties.
Steroids
; 176: 108911, 2021 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-34499930
12.
Pd-catalyzed Suzuki-Miyaura couplings and evaluation of 13α-estrone derivatives as potential anticancer agents.
Steroids
; 164: 108731, 2020 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-32946911
13.
Structural dissection of 13-epiestrones based on the interaction with human Organic anion-transporting polypeptide, OATP2B1.
J Steroid Biochem Mol Biol
; 200: 105652, 2020 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-32147459
14.
Phenolic composition and antioxidant activity of colored oats.
Food Chem
; 268: 153-161, 2018 Dec 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-30064743
15.
Synthesis of A-ring halogenated 13α-estrone derivatives as potential 17ß-HSD1 inhibitors.
Steroids
; 104: 230-6, 2015 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-26476182
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