Detalles de la búsqueda
1.
Synthesis and evaluation of antibody-drug conjugates with high drug-to-antibody ratio using dimaleimide-DM1 as a linker- payload.
Bioorg Chem
; 149: 107504, 2024 Aug.
Artículo
en Inglés
| MEDLINE | ID: mdl-38850783
2.
Analytical Method Development for 19 Alkyl Halides as Potential Genotoxic Impurities by Analytical Quality by Design.
Molecules
; 27(14)2022 Jul 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-35889310
3.
Structure-Activity Relationship Studies Based on 3D-QSAR CoMFA/CoMSIA for Thieno-Pyrimidine Derivatives as Triple Negative Breast Cancer Inhibitors.
Molecules
; 27(22)2022 Nov 17.
Artículo
en Inglés
| MEDLINE | ID: mdl-36432075
4.
Polymethoxyselenoflavones exert anti-obesity effects through activation of lipolysis and brown adipocyte metabolism.
Int J Obes (Lond)
; 45(1): 122-129, 2021 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-32467614
5.
Nordihydroguaiaretic Acid as a Novel Substrate and Inhibitor of Catechol O-Methyltransferase Modulates 4-Hydroxyestradiol-Induced Cyto- and Genotoxicity in MCF-7 Cells.
Molecules
; 26(7)2021 Apr 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-33916785
6.
Rational design of small molecule RHOA inhibitors for gastric cancer.
Pharmacogenomics J
; 20(4): 601-612, 2020 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-32015453
7.
Differential effects, on oncogenic pathway signalling, by derivatives of the HNF4 α inhibitor BI6015.
Br J Cancer
; 120(5): 488-498, 2019 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-30792535
8.
Benzo[b]tellurophenes as a Potential Histone H3 Lysine 9 Demethylase (KDM4) Inhibitor.
Int J Mol Sci
; 20(23)2019 Nov 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-31775247
9.
Efficient synthesis of polymethoxyselenoflavones via regioselective direct C-H arylation of selenochromones.
Org Biomol Chem
; 15(14): 3074-3083, 2017 Apr 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-28321447
10.
Effective and novel enantioselective preparation of pyranopyrazoles and pyranocoumarins that is catalyzed by a quinine-derived primary amine.
Org Biomol Chem
; 14(2): 623-630, 2016 Jan 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-26540619
11.
Synthesis and Evaluation of Neuroprotective Selenoflavanones.
Int J Mol Sci
; 16(12): 29574-82, 2015 Dec 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-26690420
12.
A novel synthetic compound 4-acetyl-3-methyl-6-(2-bromophenyl)pyrano[3,4-c]pyran-1,8-dione inhibits the production of nitric oxide and proinflammatory cytokines via the NF-κB pathway in lipopolysaccharide-activated microglia cells.
Neurochem Res
; 38(4): 807-14, 2013 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-23377856
13.
A synthetic compound, 4-acetyl-3-methyl-6-(3,4,5-trimethoxyphenyl)pyrano[3,4-c]pyran-1,8-dione, ameliorates ovalbumin-induced asthma.
Bioorg Med Chem
; 21(21): 6359-65, 2013 Nov 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-24054491
14.
Melittin derived peptide-drug conjugate, M-DM1, inhibits tumor progression and induces effector cell infiltration in melanoma by targeting M2 tumor-associated macrophages.
Front Immunol
; 14: 1178776, 2023.
Artículo
en Inglés
| MEDLINE | ID: mdl-37122692
15.
Distribution and Control of Bacterial Community Composition in Marian Cove Surface Waters, King George Island, Antarctica during the Summer of 2018.
Microorganisms
; 8(8)2020 Jul 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-32722258
16.
Endogenous hydrogen peroxide regulates glutathione redox via nuclear factor erythroid 2-related factor 2 downstream of phosphatidylinositol 3-kinase during muscle differentiation.
Am J Pathol
; 172(6): 1529-41, 2008 Jun.
Artículo
en Inglés
| MEDLINE | ID: mdl-18458092
17.
Synthesis of biflavones having a 6-O-7'' linkage and effects on cyclooxygenase-2 and inducible nitric oxide synthase.
Bioorg Med Chem Lett
; 19(1): 74-6, 2009 Jan 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-19041241
18.
Anti-proliferative and apoptosis induction activity of green tea polyphenols on human promyelocytic leukemia HL-60 cells.
Anticancer Res
; 29(4): 1417-21, 2009 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-19414396
19.
Bis-(3-hydroxyphenyl) diselenide inhibits LPS-stimulated iNOS and COX-2 expression in RAW 264.7 macrophage cells through the NF-kappaB inactivation.
J Pharm Pharmacol
; 61(4): 479-86, 2009 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-19298695
20.
Estrogen Receptor-Mediated Transcriptional Activities of Spent Coffee Grounds and Spent Coffee Grounds Compost, and Their Phenolic Acid Constituents.
J Agric Food Chem
; 67(31): 8649-8659, 2019 Aug 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-31283213