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1.
Structural basis for activation of fungal sterol receptor Upc2 and azole resistance.
Nat Chem Biol
; 18(11): 1253-1262, 2022 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-36229681
2.
Novel innovative computer-based test (Inno-CBT) item types for national licensing examinations for health care professionals.
BMC Med Educ
; 23(1): 560, 2023 Aug 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-37559039
3.
6'-ß-Fluoro-Homoaristeromycin and 6'-Fluoro-Homoneplanocin A Are Potent Inhibitors of Chikungunya Virus Replication through Their Direct Effect on Viral Nonstructural Protein 1.
Antimicrob Agents Chemother
; 64(4)2020 03 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-31964798
4.
Structure-Activity Relationships of Acyclic Selenopurine Nucleosides as Antiviral Agents.
Molecules
; 22(7)2017 Jul 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-28704950
5.
Asymmetric total synthesis of (+)-bermudenynol, a C15 Laurencia metabolite with a vinyl chloride containing oxocene skeleton, through intramolecular amide enolate alkylation.
Angew Chem Int Ed Engl
; 53(1): 272-6, 2014 Jan 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-24227662
6.
A novel FGFR1 inhibitor CYY292 suppresses tumor progression, invasion, and metastasis of glioblastoma by inhibiting the Akt/GSK3ß/snail signaling axis.
Genes Dis
; 11(1): 479-494, 2024 Jan.
Artículo
en Inglés
| MEDLINE | ID: mdl-37588207
7.
Corrigendum to "A novel FGFR1 inhibitor CYY292 suppresses tumor progression, invasion, and metastasis of glioblastoma by inhibiting the Akt/GSK3ß/snail signaling axis" [Genes & Diseases 11 (2024) 479-494].
Genes Dis
; 11(3): 101168, 2024 May.
Artículo
en Inglés
| MEDLINE | ID: mdl-38292171
8.
Structural Modification and Biological Evaluation of 2,8-Disubstituted Adenine and Its Nucleosides as A2A Adenosine Receptor Antagonists: Exploring the Roles of Ribose at Adenosine Receptors.
J Med Chem
; 2024 Jun 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-38845345
9.
Design and Synthesis of l-1'-Homologated Adenosine Derivatives as Potential Anti-inflammatory Agents.
ACS Omega
; 8(39): 36361-36369, 2023 Oct 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-37810713
10.
Synthesis of 9-Cinnamyl-9H-purine Derivatives as Novel TLR4/MyD88/NF-κB Pathway Inhibitors for Anti-inflammatory Effects.
ACS Med Chem Lett
; 14(12): 1839-1847, 2023 Dec 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-38116448
11.
In Silico Discovery of 5'-Modified 7-Deoxy-7-ethynyl-4'-thioadenosine as a HASPIN Inhibitor and Its Synergistic Anticancer Effect with the PLK1 Inhibitor.
ACS Cent Sci
; 9(6): 1140-1149, 2023 Jun 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-37396870
12.
Structure-Activity Relationships of Truncated 1'-Homologated Carbaadenosine Derivatives as New PPARγ/δ Ligands: A Study on Sugar Puckering Affecting Binding to PPARs.
J Med Chem
; 66(7): 4961-4978, 2023 04 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-36967575
13.
Structure-Activity Relationship of Truncated 2,8-Disubstituted-Adenosine Derivatives as Dual A2A/A3 Adenosine Receptor Antagonists and Their Cancer Immunotherapeutic Activity.
J Med Chem
; 66(17): 12249-12265, 2023 09 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-37603705
14.
Synthesis of Enantiomerically Pure Pyrimidine Ribonucleosides Locked in the South Conformation.
Org Lett
; 24(50): 9281-9284, 2022 12 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-36512445
15.
Design, Synthesis, and Biological Activity of l-1'-Homologated Adenosine Derivatives.
ACS Med Chem Lett
; 13(7): 1131-1136, 2022 Jul 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-35859875
16.
GPCR Agonist-to-Antagonist Conversion: Enabling the Design of Nucleoside Functional Switches for the A2A Adenosine Receptor.
J Med Chem
; 65(17): 11648-11657, 2022 09 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-35977382
17.
Development of a Potent Brain-Penetrant EGFR Tyrosine Kinase Inhibitor against Malignant Brain Tumors.
ACS Med Chem Lett
; 11(10): 1799-1809, 2020 Oct 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-33062157
18.
Identification of 6'-ß-fluoro-homoaristeromycin as a potent inhibitor of chikungunya virus replication.
Eur J Med Chem
; 187: 111956, 2020 Feb 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-31841728
19.
Discovery and Structure-Activity Relationships of Novel Template, Truncated 1'-Homologated Adenosine Derivatives as Pure Dual PPARγ/δ Modulators.
J Med Chem
; 63(24): 16012-16027, 2020 12 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-33325691
20.
Synthesis and anti-HIV activity of L-2',3'-Dideoxy-4'-selenonucleosides (L-4'-Se-ddNs).
Arch Pharm Res
; 42(9): 780-789, 2019 Sep.
Artículo
en Inglés
| MEDLINE | ID: mdl-31041687