Detalles de la búsqueda
1.
A hit expansion of 3-benzamidopyrazine-2-carboxamide: Toward inhibitors of prolyl-tRNA synthetase with antimycobacterial activity.
Arch Pharm (Weinheim)
; : e2400171, 2024 May 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-38710636
2.
Design, Synthesis and Antimicrobial Evaluation of New N-(1-Hydroxy-1,3-dihydrobenzo[c][1,2]oxaborol-6-yl)(hetero)aryl-2-carboxamides as Potential Inhibitors of Mycobacterial Leucyl-tRNA Synthetase.
Int J Mol Sci
; 24(3)2023 Feb 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-36769275
3.
Design of semisynthetic derivatives of the Amaryllidaceae alkaloid ambelline and exploration of their in vitro cytotoxic activities.
Saudi Pharm J
; 31(8): 101684, 2023 Aug.
Artículo
en Inglés
| MEDLINE | ID: mdl-37457365
4.
Reaction Outcome Critically Dependent on the Method of Workup: An Example from the Synthesis of 1-Isoquinolones.
J Org Chem
; 86(12): 8078-8088, 2021 Jun 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-34032448
5.
Huprine Y - Tryptophan heterodimers with potential implication to Alzheimer's disease treatment.
Bioorg Med Chem Lett
; 43: 128100, 2021 07 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-33984470
6.
Derivatives of montanine-type alkaloids and their implication for the treatment of Alzheimer's disease: Synthesis, biological activity and in silico study.
Bioorg Med Chem Lett
; 51: 128374, 2021 11 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-34555506
7.
Alkaloids of Zephyranthes citrina (Amaryllidaceae) and their implication to Alzheimer's disease: Isolation, structural elucidation and biological activity.
Bioorg Chem
; 107: 104567, 2021 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-33387730
8.
Amaryllidaceae Alkaloids of Norbelladine-Type as Inspiration for Development of Highly Selective Butyrylcholinesterase Inhibitors: Synthesis, Biological Activity Evaluation, and Docking Studies.
Int J Mol Sci
; 22(15)2021 Aug 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-34361074
9.
Semisynthetic Derivatives of Selected Amaryllidaceae Alkaloids as a New Class of Antimycobacterial Agents.
Molecules
; 26(19)2021 Oct 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-34641567
10.
Structure Elucidation and Cholinesterase Inhibition Activity of Two New Minor Amaryllidaceae Alkaloids.
Molecules
; 26(5)2021 Feb 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-33652925
11.
Aromatic Esters of the Crinane Amaryllidaceae Alkaloid Ambelline as Selective Inhibitors of Butyrylcholinesterase.
J Nat Prod
; 83(5): 1359-1367, 2020 05 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-32309949
12.
Functionalized aromatic esters of the Amaryllidaceae alkaloid haemanthamine and their in vitro and in silico biological activity connected to Alzheimer's disease.
Bioorg Chem
; 100: 103928, 2020 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-32450384
13.
N-Pyrazinoyl Substituted Amino Acids as Potential Antimycobacterial Agents-The Synthesis and Biological Evaluation of Enantiomers.
Molecules
; 25(7)2020 Mar 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-32230728
14.
A New Insight into the Stereoelectronic Control of the Pd0 -Catalyzed Allylic Substitution: Application for the Synthesis of Multisubstituted Pyran-2-ones via an Unusual 1,3-Transposition.
Chemistry
; 25(34): 8053-8060, 2019 Jun 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-30897237
15.
Isoquinoline Alkaloids from Berberis vulgaris as Potential Lead Compounds for the Treatment of Alzheimer's Disease.
J Nat Prod
; 82(2): 239-248, 2019 02 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-30701972
16.
Derivatives of 3-Aminopyrazine-2-carboxamides: Synthesis, Antimicrobial Evaluation, and in Vitro Cytotoxicity.
Molecules
; 24(7)2019 Mar 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-30925695
17.
Design, Synthesis, and Biological Evaluation of Isothiosemicarbazones with Antimycobacterial Activity.
Arch Pharm (Weinheim)
; 350(8)2017 Aug.
Artículo
en Inglés
| MEDLINE | ID: mdl-28635184
18.
Cholinesterase and Prolyl Oligopeptidase Inhibitory Activities of Alkaloids from Argemone platyceras (Papaveraceae).
Molecules
; 22(7)2017 Jul 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-28708094
19.
Design, Synthesis, Antimycobacterial Evaluation, and In Silico Studies of 3-(Phenylcarbamoyl)-pyrazine-2-carboxylic Acids.
Molecules
; 22(9)2017 Sep 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-28880230
20.
3-Substituted N-Benzylpyrazine-2-carboxamide Derivatives: Synthesis, Antimycobacterial and Antibacterial Evaluation.
Molecules
; 22(3)2017 Mar 21.
Artículo
en Inglés
| MEDLINE | ID: mdl-28335571