Detalles de la búsqueda
1.
Sofosbuvir and its tri-phosphate metabolite inhibit the RNA-dependent RNA polymerase activity of non-structural protein 5 from the Kyasanur forest disease virus.
Biochem Biophys Res Commun
; 641: 50-56, 2023 01 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-36521285
2.
Refolding and characterization of a diabody against Pfs25, a vaccine candidate of Plasmodium falciparum.
Anal Biochem
; 655: 114830, 2022 10 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-35944694
3.
Structure-guided discovery of 2-aryl/pyridin-2-yl-1H-indole derivatives as potent and selective hepsin inhibitors.
Bioorg Med Chem Lett
; 25(22): 5309-14, 2015 Nov 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-26421993
4.
Discovery of 7-azaindole based anaplastic lymphoma kinase (ALK) inhibitors: wild type and mutant (L1196M) active compounds with unique binding mode.
Bioorg Med Chem Lett
; 23(17): 4911-8, 2013 Sep 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-23880539
5.
Plasmodium chitinases: revisiting a target of transmission-blockade against malaria.
Protein Sci
; 30(8): 1493-1501, 2021 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-33934433
6.
PD-1 derived CA-170 is an oral immune checkpoint inhibitor that exhibits preclinical anti-tumor efficacy.
Commun Biol
; 4(1): 699, 2021 06 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-34103659
7.
Ternary complex formation of AFN-1252 with Acinetobacter baumannii FabI and NADH: Crystallographic and biochemical studies.
Chem Biol Drug Des
; 96(2): 704-713, 2020 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-32227402
8.
AFN-1252 is a potent inhibitor of enoyl-ACP reductase from Burkholderia pseudomallei--Crystal structure, mode of action, and biological activity.
Protein Sci
; 24(5): 832-40, 2015 May.
Artículo
en Inglés
| MEDLINE | ID: mdl-25644789
9.
Discovery of azetidine based ene-amides as potent bacterial enoyl ACP reductase (FabI) inhibitors.
Eur J Med Chem
; 84: 382-94, 2014 Sep 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-25036796
10.
Replacement of a conserved tyrosine by tryptophan in Gal3p of Saccharomyces cerevisiae reduces constitutive activity: implications for signal transduction in the GAL regulon.
Mol Genet Genomics
; 274(4): 384-93, 2005 Nov.
Artículo
en Inglés
| MEDLINE | ID: mdl-16160853
Resultados
1 -
10
de 10
1
Próxima >
>>