Detalles de la búsqueda
1.
Uncovering the Power of GPR18 Signalling: How RvD2 and Other Ligands Could Have the Potential to Modulate and Resolve Inflammation in Various Health Disorders.
Molecules
; 29(6)2024 Mar 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-38542895
2.
Anti-inflammatory effects of new human histamine H3 receptor ligands with flavonoid structure on BV-2 neuroinflammation.
Inflamm Res
; 72(2): 181-194, 2023 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-36370200
3.
The Potent and Selective Histamine H3 Receptor Antagonist E169 Counteracts Cognitive Deficits and Mitigates Disturbances in the PI3K/AKT/GSK-3ß Signaling Pathway in MK801-Induced Amnesia in Mice.
Int J Mol Sci
; 24(16)2023 Aug 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-37628900
4.
Anti-Inflammatory Activities of 8-Benzylaminoxanthines Showing High Adenosine A2A and Dual A1/A2A Receptor Affinity.
Int J Mol Sci
; 24(18)2023 Sep 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-37762006
5.
New Triazine Derivatives as Serotonin 5-HT6 Receptor Ligands.
Molecules
; 28(3)2023 Jan 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-36770774
6.
Multitargeting Histamine H3 Receptor Ligands among Acetyl- and Propionyl-Phenoxyalkyl Derivatives.
Molecules
; 28(5)2023 Mar 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-36903593
7.
Trisubstituted 1,3,5-Triazines as Histamine H4 Receptor Antagonists with Promising Activity In Vivo.
Molecules
; 28(10)2023 May 19.
Artículo
en Inglés
| MEDLINE | ID: mdl-37241939
8.
Benzophenone Derivatives with Histamine H3 Receptor Affinity and Cholinesterase Inhibitory Potency as Multitarget-Directed Ligands for Possible Therapy of Alzheimer's Disease.
Molecules
; 28(1)2022 Dec 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-36615435
9.
Cyanobiphenyls: Novel H3 receptor ligands with cholinesterase and MAO B inhibitory activity as multitarget compounds for potential treatment of Alzheimer's disease.
Bioorg Chem
; 114: 105129, 2021 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-34217977
10.
Biphenylalkoxyamine Derivatives-Histamine H3 Receptor Ligands with Butyrylcholinesterase Inhibitory Activity.
Molecules
; 26(12)2021 Jun 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-34208297
11.
In silico and in vitro studies on interaction of novel non-imidazole histamine H3R antagonists with CYP3A4.
Bioorg Med Chem Lett
; 30(11): 127147, 2020 06 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-32249114
12.
Dual Target Ligands with 4-tert-Butylphenoxy Scaffold as Histamine H3 Receptor Antagonists and Monoamine Oxidase B Inhibitors.
Int J Mol Sci
; 21(10)2020 May 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-32408504
13.
The Dual-Active Histamine H3 Receptor Antagonist and Acetylcholine Esterase Inhibitor E100 Alleviates Autistic-Like Behaviors and Oxidative Stress in Valproic Acid Induced Autism in Mice.
Int J Mol Sci
; 21(11)2020 Jun 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-32503208
14.
Antagonism of Histamine H3 receptors Alleviates Pentylenetetrazole-Induced Kindling and Associated Memory Deficits by Mitigating Oxidative Stress, Central Neurotransmitters, and c-Fos Protein Expression in Rats.
Molecules
; 25(7)2020 Mar 30.
Artículo
en Inglés
| MEDLINE | ID: mdl-32235506
15.
Alkyl derivatives of 1,3,5-triazine as histamine H4 receptor ligands.
Bioorg Med Chem
; 27(7): 1254-1262, 2019 04 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-30792106
16.
Synthesis and computer-aided analysis of the role of linker for novel ligands of the 5-HT6 serotonin receptor among substituted 1,3,5-triazinylpiperazines.
Bioorg Chem
; 84: 319-325, 2019 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-30530073
17.
Role of Histamine H3 Receptor Antagonists on Intraocular Pressure Reduction in Rabbit Models of Transient Ocular Hypertension and Glaucoma.
Int J Mol Sci
; 20(4)2019 Feb 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-30813468
18.
The Neuroprotective Effects of Histamine H3 Receptor Antagonist E177 on Pilocarpine-Induced Status Epilepticus in Rats.
Molecules
; 24(22)2019 Nov 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-31739417
19.
Are the Hydantoin-1,3,5-triazine 5-HT6R Ligands a Hope to a Find New Procognitive and Anti-Obesity Drug? Considerations Based on Primary In Vivo Assays and ADME-Tox Profile In Vitro.
Molecules
; 24(24)2019 Dec 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-31817628
20.
4-tert-Pentylphenoxyalkyl derivatives - Histamine H3 receptor ligands and monoamine oxidase B inhibitors.
Bioorg Med Chem Lett
; 28(23-24): 3596-3600, 2018 12 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-30404719