Detalles de la búsqueda
1.
Novel guanidine derivatives targeting leukemia as selective Src/Abl dual inhibitors: Design, synthesis and anti-proliferative activity.
Bioorg Chem
; 147: 107410, 2024 Jun.
Artículo
en Inglés
| MEDLINE | ID: mdl-38688197
2.
Design, synthesis, cytotoxic activities, and molecular docking of chalcone hybrids bearing 8-hydroxyquinoline moiety with dual tubulin/EGFR kinase inhibition.
Bioorg Chem
; 134: 106444, 2023 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-36893547
3.
Development and Assessment of 1,5-Diarylpyrazole/Oxime Hybrids Targeting EGFR and JNK-2 as Antiproliferative Agents: A Comprehensive Study through Synthesis, Molecular Docking, and Evaluation.
Molecules
; 28(18)2023 Sep 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-37764297
4.
Design and synthesis of pyrimidine-5-carbonitrile hybrids as COX-2 inhibitors: Anti-inflammatory activity, ulcerogenic liability, histopathological and docking studies.
Bioorg Chem
; 108: 104555, 2021 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-33376011
5.
Design, synthesis, biological evaluation, and computational studies of novel thiazolo-pyrazole hybrids as promising selective COX-2 inhibitors: Implementation of apoptotic genes expression for ulcerogenic liability assessment.
Bioorg Chem
; 111: 104883, 2021 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-33865053
6.
Daptomycin: A Novel Macrocyclic Antibiotic as a Chiral Selector in an Organic Polymer Monolithic Capillary for the Enantioselective Analysis of a Set of Pharmaceuticals.
Molecules
; 26(12)2021 Jun 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-34207780
7.
Design, Synthesis, Biological Evaluation, and Computational Studies of Novel Tri-Aryl Imidazole-Benzene Sulfonamide Hybrids as Promising Selective Carbonic Anhydrase IX and XII Inhibitors.
Molecules
; 26(16)2021 Aug 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-34443307
8.
Synthesis, DFT Calculations, Antiproliferative, Bactericidal Activity and Molecular Docking of Novel Mixed-Ligand Salen/8-Hydroxyquinoline Metal Complexes.
Molecules
; 26(16)2021 Aug 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-34443314
9.
Design, synthesis and antiproliferative evaluation of new tricyclic fused thiazolopyrimidines targeting topoisomerase II: Molecular docking and apoptosis inducing activity.
Bioorg Chem
; 105: 104446, 2020 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-33171405
10.
Design and synthesis of new 1,6-dihydropyrimidin-2-thio derivatives targeting VEGFR-2: Molecular docking and antiproliferative evaluation.
Bioorg Chem
; 102: 104090, 2020 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-32683176
11.
Design, synthesis and molecular modeling of novel aryl carboximidamides and 3-aryl-1,2,4-oxadiazoles derived from indomethacin as potent anti-inflammatory iNOS/PGE2 inhibitors.
Bioorg Chem
; 105: 104439, 2020 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-33161252
12.
Design, synthesis and anticonvulsant activity of new imidazolidindione and imidazole derivatives.
Bioorg Chem
; 101: 104020, 2020 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-32599366
13.
Design, synthesis and antitrypanosomal activity of heteroaryl-based 1,2,4-triazole and 1,3,4-oxadiazole derivatives.
Bioorg Chem
; 100: 103933, 2020 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-32446119
14.
Tailored Tetrasubstituted Imidazole Carrying the Benzenesulfonamide Fragments as Selective Human Carbonic Anhydrase IX/XII Inhibitors.
ChemMedChem
; 19(10): e202400004, 2024 May 17.
Artículo
en Inglés
| MEDLINE | ID: mdl-38356418
15.
4-[5-(4-Chloro-phen-yl)-3-methyl-1H-pyrazol-1-yl]benzene-sulfonamide.
Acta Crystallogr Sect E Struct Rep Online
; 69(Pt 2): o295-6, 2013 Feb 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-23424563
16.
1-{(Z)-[3-(1-Hy-droxy-eth-yl)anilino]methyl-idene}naphthalen-2(1H)-one.
Acta Crystallogr Sect E Struct Rep Online
; 69(Pt 1): o106, 2013 Jan 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-23476368
17.
4-Bromo-2-[(E)-(2-fluoro-5-nitro-phenyl)iminometh-yl]phenol.
Acta Crystallogr Sect E Struct Rep Online
; 69(Pt 1): o107, 2013 Jan 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-23476369
18.
2-(4-Meth-oxy-phen-yl)-1-pentyl-4,5-di-phenyl-1H-imidazole.
Acta Crystallogr Sect E Struct Rep Online
; 69(Pt 1): o5-6, 2013 Jan 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-23476433
19.
2-[2-(4-Meth-oxy-phen-yl)-4,5-diphenyl-1H-imidazol-1-yl]ethanol.
Acta Crystallogr Sect E Struct Rep Online
; 69(Pt 4): o474-5, 2013 Apr 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-23634032
20.
2-(4-Chloro-phen-yl)-1-pentyl-4,5-di-phenyl-1H-imidazole.
Acta Crystallogr Sect E Struct Rep Online
; 69(Pt 8): o1243, 2013.
Artículo
en Inglés
| MEDLINE | ID: mdl-24109333