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1.
The potent and selective RIPK2 inhibitor BI 706039 improves intestinal inflammation in the TRUC mouse model of inflammatory bowel disease.
Am J Physiol Gastrointest Liver Physiol
; 321(5): G500-G512, 2021 11 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-34494462
2.
Optimized Target Residence Time: Typeâ I1/2 Inhibitors for p38α MAP Kinase with Improved Binding Kinetics through Direct Interaction with the R-Spine.
Angew Chem Int Ed Engl
; 56(19): 5363-5367, 2017 05 02.
Artículo
en Inglés
| MEDLINE | ID: mdl-28397331
3.
Monitoring ligand-induced conformational changes for the identification of estrogen receptor agonists and antagonists.
Angew Chem Int Ed Engl
; 54(14): 4379-82, 2015 Mar 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-25664555
4.
Effects of a long-acting secretin peptide analog alone and in combination with a GLP-1R agonist in a diet-induced obesity mouse model.
Mol Metab
; 74: 101765, 2023 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-37390979
5.
Effects of GPR139 agonism on effort expenditure for food reward in rodent models: Evidence for pro-motivational actions.
Neuropharmacology
; 213: 109078, 2022 08 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-35561791
6.
Design, Synthesis, and Biological Evaluation of Novel Type I1/2 p38α MAP Kinase Inhibitors with Excellent Selectivity, High Potency, and Prolonged Target Residence Time by Interfering with the R-Spine.
J Med Chem
; 60(19): 8027-8054, 2017 10 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-28834431
7.
Targeting Drug Resistance in EGFR with Covalent Inhibitors: A Structure-Based Design Approach.
J Med Chem
; 58(17): 6844-63, 2015 Sep 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-26275028
8.
Dibenzosuberones as p38 mitogen-activated protein kinase inhibitors with low ATP competitiveness and outstanding whole blood activity.
J Med Chem
; 56(1): 241-53, 2013 Jan 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-23270382
9.
Targeting the hinge glycine flip and the activation loop: novel approach to potent p38α inhibitors.
J Med Chem
; 55(17): 7862-74, 2012 Sep 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-22897496
10.
Targeting GSK3 from Ustilago maydis: type-II kinase inhibitors as potential antifungals.
ACS Chem Biol
; 7(7): 1257-67, 2012 Jul 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-22545924
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