Detalles de la búsqueda
1.
Synthesis of Estrone Heterodimers and Evaluation of Their In Vitro Antiproliferative Activity.
Int J Mol Sci
; 25(8)2024 Apr 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-38673860
2.
Synthesis and in vitro photodynamic activity of aza-BODIPY-based photosensitizers.
Org Biomol Chem
; 21(29): 6018-6027, 2023 07 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-37436113
3.
Investigation of the Antineoplastic Effects of 2-(4-Chlorophenyl)-13α-Estrone Sulfamate against the HPV16-Positive Human Invasive Cervical Carcinoma Cell Line SiHa.
Int J Mol Sci
; 24(7)2023 Apr 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-37047597
4.
Antiproliferative and Antimetastatic Properties of 16-Azidomethyl Substituted 3-O-Benzyl Estrone Analogs.
Int J Mol Sci
; 24(18)2023 Sep 06.
Artículo
en Inglés
| MEDLINE | ID: mdl-37762056
5.
Synthesis and Antiproliferative Activity of Steroidal Diaryl Ethers.
Molecules
; 28(3)2023 Jan 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-36770863
6.
Selective antiproliferative effect of C-2 halogenated 13α-estrones on cells expressing Organic anion-transporting polypeptide 2B1 (OATP2B1).
Toxicol Appl Pharmacol
; 429: 115704, 2021 10 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-34474082
7.
Data-Driven Ensemble Docking to Map Molecular Interactions of Steroid Analogs with Hepatic Organic Anion Transporting Polypeptides.
J Chem Inf Model
; 61(6): 3109-3127, 2021 06 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-34105971
8.
Design, synthesis and biological evaluation of novel estrone phosphonates as high affinity organic anion-transporting polypeptide 2B1 (OATP2B1) inhibitors.
Bioorg Chem
; 112: 104914, 2021 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-33932771
9.
Synthesis and evaluation of AKR1C inhibitory properties of A-ring halogenated oestrone derivatives.
J Enzyme Inhib Med Chem
; 36(1): 1500-1508, 2021 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-34227437
10.
Microwave-assisted Phospha-Michael addition reactions in the 13α-oestrone series and in vitro antiproliferative properties.
J Enzyme Inhib Med Chem
; 36(1): 1931-1937, 2021 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-34445919
11.
Transition metal-catalysed A-ring C-H activations and C(sp2)-C(sp2) couplings in the 13α-oestrone series and in vitro evaluation of antiproliferative properties.
J Enzyme Inhib Med Chem
; 36(1): 895-902, 2021 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-33771084
12.
Synthesis and evaluation of anticancer activities of 2- or 4-substituted 3-(N-benzyltriazolylmethyl)-13α-oestrone derivatives.
J Enzyme Inhib Med Chem
; 36(1): 58-67, 2021 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-33121276
13.
Synthesis of substituted 15ß-alkoxy estrone derivatives and their cofactor-dependent inhibitory effect on 17ß-HSD1.
J Enzyme Inhib Med Chem
; 34(1): 1271-1286, 2019 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-31307240
14.
Synthesis, Biological Evaluation and Docking Studies of 13-Epimeric 10-fluoro- and 10-Chloroestra-1,4-dien-3-ones as Potential Aromatase Inhibitors.
Molecules
; 24(9)2019 May 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-31072017
15.
Synthesis and structure-activity relationships of 2- and/or 4-halogenated 13ß- and 13α-estrone derivatives as enzyme inhibitors of estrogen biosynthesis.
J Enzyme Inhib Med Chem
; 33(1): 1271-1282, 2018 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-30230387
16.
Synthesis of Novel C-2- or C-15-Labeled BODIPY-Estrone Conjugates.
Molecules
; 23(4)2018 Apr 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-29614041
17.
The first Pd-catalyzed Buchwald-Hartwig aminations at C-2 or C-4 in the estrone series.
Beilstein J Org Chem
; 14: 998-1003, 2018.
Artículo
en Inglés
| MEDLINE | ID: mdl-29977371
18.
Pd-Catalyzed microwave-assisted synthesis of phosphonated 13α-estrones as potential OATP2B1, 17ß-HSD1 and/or STS inhibitors.
Beilstein J Org Chem
; 14: 2838-2845, 2018.
Artículo
en Inglés
| MEDLINE | ID: mdl-30498534
19.
Synthesis and in vitro investigation of potential antiproliferative monosaccharide-d-secoestrone bioconjugates.
Bioorg Med Chem Lett
; 27(9): 1938-1942, 2017 05 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-28343874
20.
Synthesis of novel 13α-estrone derivatives by Sonogashira coupling as potential 17ß-HSD1 inhibitors.
Beilstein J Org Chem
; 13: 1303-1309, 2017.
Artículo
en Inglés
| MEDLINE | ID: mdl-28694873