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1.
Stereoselective synthesis of 3,4-dihydropyrrolo[1,2-a]pyrazin-1(2H)-one derivatives as PIM kinase inhibitors inspired from marine alkaloids.
Chirality
; 34(11): 1437-1452, 2022 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-35959859
2.
Discovery and optimization of pyrrolo[1,2-a]pyrazinones leads to novel and selective inhibitors of PIM kinases.
Bioorg Med Chem
; 21(23): 7364-80, 2013 Dec 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-24139169
3.
The Novel PIM1 Inhibitor NMS-P645 Reverses PIM1-Dependent Effects on TMPRSS2/ERG Positive Prostate Cancer Cells And Shows Anti-Proliferative Activity in Combination with PI3K Inhibition.
J Cancer
; 8(1): 140-145, 2017.
Artículo
en Inglés
| MEDLINE | ID: mdl-28123608
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