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1.
High Throughput Combinatorial Formatting of PcrV Nanobodies for Efficient Potency Improvement.
J Biol Chem
; 291(29): 15243-55, 2016 07 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-27226529
2.
Synthesis, ligand-receptor modeling studies and pharmacological evaluation of novel 4-modified-2-aryl-1,2,4-triazolo[4,3-a]quinoxalin-1-one derivatives as potent and selective human A3 adenosine receptor antagonists.
Bioorg Med Chem
; 16(11): 6086-102, 2008 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-18468446
3.
New 2-arylpyrazolo[3,4-c]quinoline derivatives as potent and selective human A3 adenosine receptor antagonists. Synthesis, pharmacological evaluation, and ligand-receptor modeling studies.
J Med Chem
; 50(17): 4061-74, 2007 Aug 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-17665891
4.
Scouting human A3 adenosine receptor antagonist binding mode using a molecular simplification approach: from triazoloquinoxaline to a pyrimidine skeleton as a key study.
J Med Chem
; 50(26): 6596-606, 2007 Dec 27.
Artículo
en Inglés
| MEDLINE | ID: mdl-18047262
5.
4-amido-2-aryl-1,2,4-triazolo[4,3-a]quinoxalin-1-ones as new potent and selective human A3 adenosine receptor antagonists. synthesis, pharmacological evaluation, and ligand-receptor modeling studies.
J Med Chem
; 49(13): 3916-25, 2006 Jun 29.
Artículo
en Inglés
| MEDLINE | ID: mdl-16789747
6.
Human A3 adenosine receptor as versatile G protein-coupled receptor example to validate the receptor homology modeling technology.
Curr Pharm Des
; 15(35): 4069-84, 2009.
Artículo
en Inglés
| MEDLINE | ID: mdl-20028322
7.
2-Phenylpyrazolo[4,3-d]pyrimidin-7-one as a new scaffold to obtain potent and selective human A3 adenosine receptor antagonists: new insights into the receptor-antagonist recognition.
J Med Chem
; 52(23): 7640-52, 2009 Dec 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-19743865
8.
Pyrido[2,3-e]-1,2,4-triazolo[4,3-a]pyrazin-1-one as a new scaffold to develop potent and selective human A3 adenosine receptor antagonists. Synthesis, pharmacological evaluation, and ligand-receptor modeling studies.
J Med Chem
; 52(8): 2407-19, 2009 Apr 23.
Artículo
en Inglés
| MEDLINE | ID: mdl-19301821
9.
Pyrazolo-triazolo-pyrimidines as adenosine receptor antagonists: Effect of the N-5 bond type on the affinity and selectivity at the four adenosine receptor subtypes.
Purinergic Signal
; 4(1): 39-46, 2008 Mar.
Artículo
en Inglés
| MEDLINE | ID: mdl-18368532
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