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1.
Sphingosine 1-phosphate lyase inhibition by 2-acetyl-4-(tetrahydroxybutyl)imidazole (THI) under conditions of vitamin B6 deficiency.
Mol Cell Biochem
; 400(1-2): 125-33, 2015 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-25381637
2.
A novel inhibitor of I-kappaB kinase beta ameliorates experimental arthritis through downregulation of proinflammatory cytokines in arthritic joints.
Biol Pharm Bull
; 37(1): 87-95, 2014.
Artículo
en Inglés
| MEDLINE | ID: mdl-24389485
3.
A novel, potent, and orally active VLA-4 antagonist with good aqueous solubility: trans-4-[1-[[2-(5-Fluoro-2-methylphenylamino)-7-fluoro-6-benzoxazolyl]acetyl]-(5S)-[methoxy(methyl)amino]methyl-(2S)-pyrrolidinylmethoxy]cyclohexanecarboxylic acid.
Bioorg Med Chem
; 21(1): 42-61, 2013 Jan 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-23218775
4.
Identification of trans-4-[1-[[7-fluoro-2-(1-methyl-3-indolyl)-6-benzoxazolyl]acetyl]-(4S)-fluoro-(2S)-pyrrolidinylmethoxy]cyclohexanecarboxylic acid as a potent, orally active VLA-4 antagonist.
Bioorg Med Chem
; 20(3): 1201-12, 2012 Feb 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-22261021
5.
A concise synthesis of a very late antigen-4 antagonist trans-4-[1-[[2,5-dichloro-4-(1-methyl-3-indolylcarboxyamide)phenyl]acetyl]-(4S)-methoxy-(2S)-pyrrolidinylmethoxy]cyclohexanecarboxylic acid via reductive etherification.
Chem Pharm Bull (Tokyo)
; 60(7): 882-6, 2012.
Artículo
en Inglés
| MEDLINE | ID: mdl-22790822
6.
Discovery of imidazo[1,2-b]pyridazines as IKKß inhibitors. Part 3: exploration of effective compounds in arthritis models.
Bioorg Med Chem Lett
; 21(15): 4550-5, 2011 Aug 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-21705219
7.
Potent priming by inactivated whole influenza virus particle vaccines is linked to viral RNA uptake into antigen presenting cells.
Vaccine
; 39(29): 3940-3951, 2021 06 29.
Artículo
en Inglés
| MEDLINE | ID: mdl-34090697
8.
A novel and potent VLA-4 antagonist based on trans-4-substituted cyclohexanecarboxylic acid.
Bioorg Med Chem
; 17(3): 1232-43, 2009 Feb 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-19124247
9.
Identification of 4-[1-[3-chloro-4-[N'-(5-fluoro-2-methylphenyl)ureido]phenylacetyl]-(4S)-fluoro-(2S)-pyrrolidinylmethoxy]benzoic acid as a potent, orally active VLA-4 antagonist.
Bioorg Med Chem
; 16(23): 9991-10000, 2008 Dec 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-18952443
10.
Scintillation Proximity Assay to Detect the Changes in Cellular Dihydrosphingosine 1-Phosphate Levels.
Lipids
; 51(10): 1207-1216, 2016 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-27585475
11.
Component of Caramel Food Coloring, THI, Causes Lymphopenia Indirectly via a Key Metabolic Intermediate.
Cell Chem Biol
; 23(5): 555-560, 2016 05 19.
Artículo
en Inglés
| MEDLINE | ID: mdl-27185637
12.
Discovery of trans-4-[1-[[2,5-Dichloro-4-(1-methyl-3-indolylcarboxamido)phenyl]acetyl]-(4S)-methoxy-(2S)-pyrrolidinylmethoxy]cyclohexanecarboxylic acid: an orally active, selective very late antigen-4 antagonist.
J Med Chem
; 52(24): 7974-92, 2009 Dec 24.
Artículo
en Inglés
| MEDLINE | ID: mdl-19891440
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