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1.
Comparison of the effect of surgical versus transcatheter aortic valve replacement on the development of postoperative acute kidney injury.
Heart Vessels
; 39(4): 359-364, 2024 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-37978052
2.
Genome-Wide Association Study Identifies Genetic Polymorphisms Associated with Estimated Minimum Effective Concentration of Fentanyl in Patients Undergoing Laparoscopic-Assisted Colectomy.
Int J Mol Sci
; 24(9)2023 May 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-37176129
3.
Efficient synthesis of tert-butyl 3-cyano-3-cyclopropyl-2-oxopyrrolidine-4-carboxylates: Highly functionalized 2-pyrrolidinone enabling access to novel macrocyclic Tyk2 inhibitors.
Bioorg Med Chem Lett
; 30(5): 126963, 2020 03 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-31980341
4.
Vocal cord inflammatory myofibroblastic tumor with mucoid deposits harboring TIMP3-ALK fusion: A potential diagnostic pitfall.
Pathol Int
; 69(6): 366-371, 2019 Jun.
Artículo
en Inglés
| MEDLINE | ID: mdl-31215130
5.
Identification of novel quinazolinedione derivatives as RORγt inverse agonist.
Bioorg Med Chem
; 26(3): 721-736, 2018 02 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-29342416
6.
Discovery of orally efficacious RORγt inverse agonists, part 1: Identification of novel phenylglycinamides as lead scaffolds.
Bioorg Med Chem
; 26(2): 483-500, 2018 01 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-29262987
7.
Discovery of orally efficacious RORγt inverse agonists. Part 2: Design, synthesis, and biological evaluation of novel tetrahydroisoquinoline derivatives.
Bioorg Med Chem
; 26(2): 470-482, 2018 01 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-29258712
8.
Biochemical Properties of TAK-828F, a Potent and Selective Retinoid-Related Orphan Receptor Gamma t Inverse Agonist.
Pharmacology
; 102(5-6): 244-252, 2018.
Artículo
en Inglés
| MEDLINE | ID: mdl-30134246
9.
Cancer with low cathepsin D levels is susceptible to vacuolar (H+ )-ATPase inhibition.
Cancer Sci
; 108(6): 1185-1193, 2017 Jun.
Artículo
en Inglés
| MEDLINE | ID: mdl-28317223
10.
A potent and selective natriuretic peptide receptor-3 blocker 11-mer peptide created by hybridization of musclin and atrial natriuretic peptide.
Bioorg Med Chem Lett
; 27(15): 3542-3545, 2017 08 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-28596054
11.
Practical application of 3-substituted-2,6-difluoropyridines in drug discovery: Facile synthesis of novel protein kinase C theta inhibitors.
Bioorg Med Chem Lett
; 27(11): 2497-2501, 2017 06 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-28400232
12.
Discovery of 4-chloro-2-(2,4-dichloro-6-methylphenoxy)-1-methyl-7-(pentan-3-yl)-1H-benzimidazole, a novel CRF1 receptor antagonist.
Bioorg Med Chem
; 25(5): 1556-1570, 2017 03 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-28174066
13.
Design, synthesis, and biological evaluation of a novel series of peripheral-selective noradrenaline reuptake inhibitors-Part 2.
Bioorg Med Chem
; 24(14): 3207-17, 2016 07 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-27255177
14.
Design, synthesis, and biological evaluation of a novel series of peripheral-selective noradrenaline reuptake inhibitors - Part 3.
Bioorg Med Chem
; 24(16): 3716-26, 2016 08 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-27325446
15.
Discovery and optimization of 1,7-disubstituted-2,2-dimethyl-2,3-dihydroquinazolin-4(1H)-ones as potent and selective PKCθ inhibitors.
Bioorg Med Chem
; 24(11): 2466-75, 2016 06 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-27117263
16.
Fe K-Edge X-ray Absorption Fine Structure Determination of γ-Al2 O3 -Supported Iron-Oxide Species.
Chemphyschem
; 16(9): 2015-20, 2015 Jun 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-25914350
17.
Design, synthesis and biological evaluation of a novel series of peripheral-selective noradrenaline reuptake inhibitor.
Bioorg Med Chem
; 23(15): 5000-5014, 2015 Aug 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-26051602
18.
Effects of antihistamine on up-regulation of histamine H1 receptor mRNA in the nasal mucosa of patients with pollinosis induced by controlled cedar pollen challenge in an environmental exposure unit.
J Pharmacol Sci
; 129(3): 183-7, 2015 Nov.
Artículo
en Inglés
| MEDLINE | ID: mdl-26598006
19.
Design, synthesis, and biological activities of 1-aryl-1,4-diazepan-2-one derivatives as novel triple reuptake inhibitors.
Bioorg Med Chem Lett
; 24(16): 3898-902, 2014 Aug 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-25017029
20.
Novel triple reuptake inhibitors with low risk of CAD associated liabilities: design, synthesis and biological activities of 4-[(1S)-1-(3,4-dichlorophenyl)-2-methoxyethyl]piperidine and related compounds.
Bioorg Med Chem
; 21(15): 4600-13, 2013 Aug 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-23769168