Detalles de la búsqueda
1.
Derivatization of inhibitor of apoptosis protein (IAP) ligands yields improved inducers of estrogen receptor α degradation.
J Biol Chem
; 293(18): 6776-6790, 2018 05 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-29545311
2.
Different Degradation Mechanisms of Inhibitor of Apoptosis Proteins (IAPs) by the Specific and Nongenetic IAP-Dependent Protein Eraser (SNIPER).
Chem Pharm Bull (Tokyo)
; 67(3): 203-209, 2019 Mar 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-30369550
3.
In Vivo Knockdown of Pathogenic Proteins via Specific and Nongenetic Inhibitor of Apoptosis Protein (IAP)-dependent Protein Erasers (SNIPERs).
J Biol Chem
; 292(11): 4556-4570, 2017 03 17.
Artículo
en Inglés
| MEDLINE | ID: mdl-28154167
4.
SNIPER(TACC3) induces cytoplasmic vacuolization and sensitizes cancer cells to Bortezomib.
Cancer Sci
; 108(5): 1032-1041, 2017 May.
Artículo
en Inglés
| MEDLINE | ID: mdl-28192613
5.
Development of protein degradation inducers of oncogenic BCR-ABL protein by conjugation of ABL kinase inhibitors and IAP ligands.
Cancer Sci
; 108(8): 1657-1666, 2017 Aug.
Artículo
en Inglés
| MEDLINE | ID: mdl-28556300
6.
Design, synthesis, and biological activity of novel, potent, and highly selective fused pyrimidine-2-carboxamide-4-one-based matrix metalloproteinase (MMP)-13 zinc-binding inhibitors.
Bioorg Med Chem
; 24(23): 6149-6165, 2016 12 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-27825552
7.
Thieno[2,3-d]pyrimidine-2-carboxamides bearing a carboxybenzene group at 5-position: highly potent, selective, and orally available MMP-13 inhibitors interacting with the S1â³ binding site.
Bioorg Med Chem
; 22(19): 5487-505, 2014 Oct 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-25192810
8.
Second-Generation AUTACs for Targeted Autophagic Degradation.
J Med Chem
; 66(17): 12342-12372, 2023 09 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-37589438
9.
Pharmacological inhibition of PRMT7 links arginine monomethylation to the cellular stress response.
Nat Commun
; 11(1): 2396, 2020 05 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-32409666
10.
Author Correction: Pharmacological inhibition of PRMT7 links arginine monomethylation to the cellular stress response.
Nat Commun
; 11(1): 2683, 2020 05 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-32457299
11.
Pharmacological difference between degrader and inhibitor against oncogenic BCR-ABL kinase.
Sci Rep
; 8(1): 13549, 2018 09 10.
Artículo
en Inglés
| MEDLINE | ID: mdl-30202081
12.
Development of Protein Degradation Inducers of Androgen Receptor by Conjugation of Androgen Receptor Ligands and Inhibitor of Apoptosis Protein Ligands.
J Med Chem
; 61(2): 543-575, 2018 01 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-28594553
13.
Targeting the Allosteric Site of Oncoprotein BCR-ABL as an Alternative Strategy for Effective Target Protein Degradation.
ACS Med Chem Lett
; 8(10): 1042-1047, 2017 Oct 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-29057048
14.
Discovery of Novel, Highly Potent, and Selective Matrix Metalloproteinase (MMP)-13 Inhibitors with a 1,2,4-Triazol-3-yl Moiety as a Zinc Binding Group Using a Structure-Based Design Approach.
J Med Chem
; 60(2): 608-626, 2017 01 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-27966948
15.
Discovery of novel, highly potent, and selective quinazoline-2-carboxamide-based matrix metalloproteinase (MMP)-13 inhibitors without a zinc binding group using a structure-based design approach.
J Med Chem
; 57(21): 8886-902, 2014 Nov 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-25264600
Resultados
1 -
15
de 15
1
Próxima >
>>