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1.
Optimizing and characterizing 4-methyl substituted pyrazol-3-carboxamides leading to the peripheral cannabinoid 1 receptor inverse agonist TM38837.
Bioorg Med Chem Lett
; 98: 129572, 2024 Jan 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-38043690
2.
A novel GIP analogue, ZP4165, enhances glucagon-like peptide-1-induced body weight loss and improves glycaemic control in rodents.
Diabetes Obes Metab
; 20(1): 60-68, 2018 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-28598027
3.
Efficacy in diet-induced obese mice of the hepatotropic, peripheral cannabinoid 1 receptor inverse agonist TM38837.
Br J Pharmacol
; 2024 Jun 17.
Artículo
en Inglés
| MEDLINE | ID: mdl-38886096
4.
Exploring SAR features in diverse library of 4-cyanomethyl-pyrazole-3-carboxamides suitable for further elaborations as CB1 antagonists.
Bioorg Med Chem Lett
; 20(1): 26-30, 2010 Jan 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-19954978
5.
Conversion of 4-cyanomethyl-pyrazole-3-carboxamides into CB1 antagonists with lowered propensity to pass the blood-brain-barrier.
Bioorg Med Chem Lett
; 20(2): 453-7, 2010 Jan 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-20015647
6.
6-Acylamino-2-aminoquinolines as potent melanin-concentrating hormone 1 receptor antagonists. Identification, structure-activity relationship, and investigation of binding mode.
J Med Chem
; 48(18): 5684-97, 2005 Sep 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-16134937
7.
6-Acylamino-2-amino-4-methylquinolines as potent melanin-concentrating hormone 1 receptor antagonists: structure-activity exploration of eastern and western parts.
Bioorg Med Chem Lett
; 16(4): 1070-5, 2006 Feb 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-16289819
8.
A highly conserved glycine within linker I and the extreme C terminus of G protein alpha subunits interact cooperatively in switching G protein-coupled receptor-to-effector specificity.
J Pharmacol Exp Ther
; 313(1): 78-87, 2005 Apr.
Artículo
en Inglés
| MEDLINE | ID: mdl-15615862
9.
4-Acylamino-and 4-ureidobenzamides as melanin-concentrating hormone (MCH) receptor 1 antagonists.
Bioorg Med Chem Lett
; 14(20): 5075-80, 2004 Oct 18.
Artículo
en Inglés
| MEDLINE | ID: mdl-15380202
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