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1.
Syntheses and pharmacokinetic evaluations of four metabolites of 2-(4-(2-((1H-benzo[d]imidazol-2-yl)thio)ethyl)piperazin-1-yl)-N-(6-methyl-2,4-bis-(methylthio)pyridin-3-yl)acetamide hydrochloride [K-604], an acyl-CoA:cholesterol O-acyltransferase-1 inhibitor.
Bioorg Med Chem
; 28(11): 115457, 2020 06 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-32334935
2.
Discovery of novel spiro[chromane-2,4'-piperidine] derivatives as potent and orally bioavailable G-protein-coupled receptor 119 agonists.
Bioorg Med Chem Lett
; 28(19): 3236-3241, 2018 10 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-30145005
3.
Optimization of a novel series of potent and orally bioavailable GPR119 agonists.
Bioorg Med Chem Lett
; 27(15): 3249-3253, 2017 08 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-28648463
4.
New CETP inhibitor K-312 reduces PCSK9 expression: a potential effect on LDL cholesterol metabolism.
Am J Physiol Endocrinol Metab
; 309(2): E177-90, 2015 Jul 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-26015437
5.
Three derivatives of 4-fluoro-5-sulfonylisoquinoline.
Acta Crystallogr C
; 68(Pt 10): o427-30, 2012 Oct.
Artículo
en Inglés
| MEDLINE | ID: mdl-23007548
6.
Discovery of Clinical Candidate 2-(4-(2-((1 H-Benzo[ d]imidazol-2-yl)thio)ethyl)piperazin-1-yl)- N-(6-methyl-2,4-bis(methylthio)pyridin-3-yl)acetamide Hydrochloride [K-604], an Aqueous-Soluble Acyl-CoA:Cholesterol O-Acyltransferase-1 Inhibitor.
J Med Chem
; 61(23): 10635-10650, 2018 12 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-30433781
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