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1.
Discovery of Novel Imidazopyridine GSK-3ß Inhibitors Supported by Computational Approaches.
Molecules
; 25(9)2020 May 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-32380735
2.
Structure-Based Discovery of 1H-Indazole-3-carboxamides as a Novel Structural Class of Human GSK-3 Inhibitors.
J Chem Inf Model
; 55(12): 2540-51, 2015 Dec 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-26600430
3.
Murine mPGES-1 3D structure elucidation and inhibitors binding mode predictions by homology modeling and site-directed mutagenesis.
J Chem Inf Model
; 53(7): 1804-17, 2013 Jul 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-23789712
4.
Molecular Insights Into Binding and Activation of the Human KCNQ2 Channel by Retigabine.
Front Mol Biosci
; 9: 839249, 2022.
Artículo
en Inglés
| MEDLINE | ID: mdl-35309507
5.
Testing Fmr1 KO Phenotypes in Response to GSK3 Inhibitors: SB216763 versus AFC03127.
Front Mol Neurosci
; 14: 751307, 2021.
Artículo
en Inglés
| MEDLINE | ID: mdl-34690696
6.
Discovery of Novel Chemical Series of OXA-48 ß-Lactamase Inhibitors by High-Throughput Screening.
Pharmaceuticals (Basel)
; 14(7)2021 Jun 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-34202402
7.
Structure-based virtual screening to identify novel carnitine acetyltransferase activators.
J Mol Graph Model
; 100: 107692, 2020 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-32759041
8.
The mood stabilizing properties of AF3581, a novel potent GSK-3ß inhibitor.
Biomed Pharmacother
; 128: 110249, 2020 Aug.
Artículo
en Inglés
| MEDLINE | ID: mdl-32470749
9.
Antibacterial activity of novel dual bacterial DNA type II topoisomerase inhibitors.
PLoS One
; 15(2): e0228509, 2020.
Artículo
en Inglés
| MEDLINE | ID: mdl-32074119
10.
Optimization of Indazole-Based GSK-3 Inhibitors with Mitigated hERG Issue and In Vivo Activity in a Mood Disorder Model.
ACS Med Chem Lett
; 11(5): 825-831, 2020 May 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-32435391
11.
Virtual Screening Approach and Investigation of Structure-Activity Relationships To Discover Novel Bacterial Topoisomerase Inhibitors Targeting Gram-Positive and Gram-Negative Pathogens.
J Med Chem
; 62(16): 7445-7472, 2019 08 22.
Artículo
en Inglés
| MEDLINE | ID: mdl-31276392
12.
Molecular basis for the different interactions of congeneric substrates with the polyspecific transporter AcrB.
Biochim Biophys Acta Biomembr
; 1861(7): 1397-1408, 2019 07 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-31075229
13.
New anti-viral drugs for the treatment of the common cold.
Bioorg Med Chem
; 16(6): 3091-107, 2008 Mar 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-18248816
14.
A Novel Multi-step Virtual Screening for the Identification of Human and Mouse mPGES-1 Inhibitors.
Mol Inform
; 35(8-9): 358-68, 2016 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-27546040
15.
Hit Optimization of 5-Substituted-N-(piperidin-4-ylmethyl)-1H-indazole-3-carboxamides: Potent Glycogen Synthase Kinase-3 (GSK-3) Inhibitors with in Vivo Activity in Model of Mood Disorders.
J Med Chem
; 58(22): 8920-37, 2015 Nov 25.
Artículo
en Inglés
| MEDLINE | ID: mdl-26486317
16.
Discovery and pharmacological profile of new 1H-indazole-3-carboxamide and 2H-pyrrolo[3,4-c]quinoline derivatives as selective serotonin 4 receptor ligands.
J Med Chem
; 55(22): 9446-66, 2012 Nov 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-23043420
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