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1.
Design, synthesis, and structure-activity relationships of a series of novel N-aryl-2-phenylcyclopropanecarboxamide that are potent and orally active orexin receptor antagonists.
Bioorg Med Chem
; 22(21): 6071-88, 2014 Nov 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-25267004
2.
Discovery of (1R,2S)-2-{[(2,4-Dimethylpyrimidin-5-yl)oxy]methyl}-2-(3-fluorophenyl)-N-(5-fluoropyridin-2-yl)cyclopropanecarboxamide (E2006): A Potent and Efficacious Oral Orexin Receptor Antagonist.
J Med Chem
; 58(11): 4648-64, 2015 Jun 11.
Artículo
en Inglés
| MEDLINE | ID: mdl-25953512
3.
Piperidine carboxylic acid derivatives of 10H-pyrazino[2,3-b][1,4]benzothiazine as orally-active adhesion molecule inhibitors.
Chem Pharm Bull (Tokyo)
; 52(6): 675-87, 2004 Jun.
Artículo
en Inglés
| MEDLINE | ID: mdl-15187387
4.
Inhibitors of adhesion molecules expression; the synthesis and pharmacological properties of 10H-pyrazino[2,3-b][1,4]benzothiazine derivatives.
Chem Pharm Bull (Tokyo)
; 50(7): 922-9, 2002 Jul.
Artículo
en Inglés
| MEDLINE | ID: mdl-12130850
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