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1.
An electrophoretic mobility shift assay for the identification and kinetic analysis of acetyl transferase inhibitors.
Anal Biochem
; 402(1): 65-8, 2010 Jul 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-20338149
2.
Benzo[d]imidazole inhibitors of Coactivator Associated Arginine Methyltransferase 1 (CARM1)--Hit to Lead studies.
Bioorg Med Chem Lett
; 19(17): 5063-6, 2009 Sep 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-19632837
3.
Optimization of pyrazole inhibitors of Coactivator Associated Arginine Methyltransferase 1 (CARM1).
Bioorg Med Chem Lett
; 19(11): 2924-7, 2009 Jun 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-19419866
4.
Pyrazole inhibitors of coactivator associated arginine methyltransferase 1 (CARM1).
Bioorg Med Chem Lett
; 18(15): 4438-41, 2008 Aug 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-18619839
5.
2-aminothiazole as a novel kinase inhibitor template. Structure-activity relationship studies toward the discovery of N-(2-chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)-1- piperazinyl)]-2-methyl-4-pyrimidinyl]amino)]-1,3-thiazole-5-carboxamide (dasatinib, BMS-354825) as a potent pan-Src kinase inhibitor.
J Med Chem
; 49(23): 6819-32, 2006 Nov 16.
Artículo
en Inglés
| MEDLINE | ID: mdl-17154512
6.
Imidazoquinoxaline Src-family kinase p56Lck inhibitors: SAR, QSAR, and the discovery of (S)-N-(2-chloro-6-methylphenyl)-2-(3-methyl-1-piperazinyl)imidazo- [1,5-a]pyrido[3,2-e]pyrazin-6-amine (BMS-279700) as a potent and orally active inhibitor with excellent in vivo antiinflammatory activity.
J Med Chem
; 47(18): 4517-29, 2004 Aug 26.
Artículo
en Inglés
| MEDLINE | ID: mdl-15317463
7.
Discovery of N-(2-chloro-6-methyl- phenyl)-2-(6-(4-(2-hydroxyethyl)- piperazin-1-yl)-2-methylpyrimidin-4- ylamino)thiazole-5-carboxamide (BMS-354825), a dual Src/Abl kinase inhibitor with potent antitumor activity in preclinical assays.
J Med Chem
; 47(27): 6658-61, 2004 Dec 30.
Artículo
en Inglés
| MEDLINE | ID: mdl-15615512
8.
Discovery of 2-amino-heteroaryl-benzothiazole-6-anilides as potent p56(lck) inhibitors.
Bioorg Med Chem Lett
; 13(15): 2587-90, 2003 Aug 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-12852972
9.
Molecular design, synthesis, and structure-Activity relationships leading to the potent and selective p56(lck) inhibitor BMS-243117.
Bioorg Med Chem Lett
; 13(13): 2145-9, 2003 Jul 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-12798323
10.
Discovery of novel 2-(aminoheteroaryl)-thiazole-5-carboxamides as potent and orally active Src-family kinase p56(Lck) inhibitors.
Bioorg Med Chem Lett
; 14(24): 6061-6, 2004 Dec 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-15546730
11.
Discovery and initial SAR of imidazoquinoxalines as inhibitors of the Src-family kinase p56(Lck).
Bioorg Med Chem Lett
; 12(10): 1361-4, 2002 May 20.
Artículo
en Inglés
| MEDLINE | ID: mdl-11992777
12.
Synthesis and SAR of novel imidazoquinoxaline-based Lck inhibitors: improvement of cell potency.
Bioorg Med Chem Lett
; 12(21): 3153-6, 2002 Nov 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-12372522
13.
Discovery and initial SAR of 2-amino-5-carboxamidothiazoles as inhibitors of the Src-family kinase p56(Lck).
Bioorg Med Chem Lett
; 13(22): 4007-10, 2003 Nov 17.
Artículo
en Inglés
| MEDLINE | ID: mdl-14592495
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