Detalles de la búsqueda
1.
Potent carbonic anhydrase I, II, IX and XII inhibition activity of novel primary benzenesulfonamides incorporating bis-ureido moieties.
J Enzyme Inhib Med Chem
; 38(1): 2185762, 2023 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36880350
2.
Novel benzenesulfonamide-thiouracil conjugates with a flexible N-ethyl acetamide linker as selective CA IX and CA XII inhibitors.
Arch Pharm (Weinheim)
; 356(2): e2200434, 2023 Feb.
Artículo
en Inglés
| MEDLINE | ID: mdl-36372524
3.
Synthesis, molecular modelling and QSAR study of new N-phenylacetamide-2-oxoindole benzensulfonamide conjugates as carbonic anhydrase inhibitors with antiproliferative activity.
J Enzyme Inhib Med Chem
; 37(1): 701-717, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-35168458
4.
2-Aminobenzoxazole-appended coumarins as potent and selective inhibitors of tumour-associated carbonic anhydrases.
J Enzyme Inhib Med Chem
; 37(1): 168-177, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-34894971
5.
Investigation of the carbonic anhydrase inhibitory activity of benzenesulfonamides incorporating substituted fused-pyrimidine tails.
Arch Pharm (Weinheim)
; 355(11): e2200274, 2022 Nov.
Artículo
en Inglés
| MEDLINE | ID: mdl-35972823
6.
Novel 2-substituted thioquinazoline-benzenesulfonamide derivatives as carbonic anhydrase inhibitors with potential anticancer activity.
Arch Pharm (Weinheim)
; 355(12): e2200180, 2022 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-36056903
7.
Novel triazole-sulfonamide bearing pyrimidine moieties with carbonic anhydrase inhibitory action: Design, synthesis, computational and enzyme inhibition studies.
Bioorg Med Chem Lett
; 48: 128249, 2021 09 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-34237441
8.
Anion inhibition studies of the Zn(II)-bound ι-carbonic anhydrase from the Gram-negative bacterium Burkholderia territorii.
J Enzyme Inhib Med Chem
; 36(1): 372-376, 2021 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-33390061
9.
Effect of amino acids and amines on the activity of the recombinant ι-carbonic anhydrase from the Gram-negative bacterium Burkholderia territorii.
J Enzyme Inhib Med Chem
; 36(1): 1000-1006, 2021 Dec.
Artículo
en Inglés
| MEDLINE | ID: mdl-33980103
10.
Synthesis and Inhibition Activity Study of Triazinyl-Substituted Amino(alkyl)-benzenesulfonamide Conjugates with Polar and Hydrophobic Amino Acids as Inhibitors of Human Carbonic Anhydrases I, II, IV, IX, and XII.
Int J Mol Sci
; 22(20)2021 Oct 19.
Artículo
en Inglés
| MEDLINE | ID: mdl-34681940
11.
Effect of Sulfonamides and Their Structurally Related Derivatives on the Activity of ι-Carbonic Anhydrase from Burkholderia territorii
Int J Mol Sci
; 22(2)2021 01 08.
Artículo
en Inglés
| MEDLINE | ID: mdl-33430028
12.
1,3-Diaryl Triazenes Incorporating Disulfonamides Show Both Antiproliferative Activity and Effective Inhibition of Tumor-associated Carbonic Anhydrases IX and XII.
Anticancer Agents Med Chem
; 2024 Feb 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-38362678
13.
Coumarin-pyrazoline Hybrids as Selective Inhibitors of the Tumor-associated Carbonic Anhydrase IX and XII.
Anticancer Agents Med Chem
; 23(10): 1217-1223, 2023.
Artículo
en Inglés
| MEDLINE | ID: mdl-36825712
14.
Discovery of new carbonic anhydrase IX inhibitors as anticancer agents by toning the hydrophobic and hydrophilic rims of the active site to encounter the dual-tail approach.
Eur J Med Chem
; 232: 114190, 2022 Mar 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-35182815
15.
Application of the dual-tail approach for the design and synthesis of novel Thiopyrimidine-Benzenesulfonamide hybrids as selective carbonic anhydrase inhibitors.
Eur J Med Chem
; 228: 114004, 2022 Jan 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-34847409
16.
Carbonic Anhydrase inhibitors bearing organotelluride moieties as novel agents for antitumor therapy.
Eur J Med Chem
; 244: 114811, 2022 Dec 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-36208508
17.
Binding site comparison for coumarin inhibitors and amine/amino acid activators of human carbonic anhydrases.
Eur J Med Chem
; 226: 113875, 2021 Dec 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-34634741
18.
Synthesis, Computational Studies and Assessment of in Vitro Activity of Squalene Derivatives as Carbonic Anhydrase Inhibitors.
ChemMedChem
; 15(21): 2052-2057, 2020 11 04.
Artículo
en Inglés
| MEDLINE | ID: mdl-32744806
19.
Inclusion of a 5-fluorouracil moiety in nitrogenous bases derivatives as human carbonic anhydrase IX and XII inhibitors produced a targeted action against MDA-MB-231 and T47D breast cancer cells.
Eur J Med Chem
; 190: 112112, 2020 Mar 15.
Artículo
en Inglés
| MEDLINE | ID: mdl-32044580
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