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1.
Estrogenic Activity of Tetrazole Derivatives Bearing Bisphenol Structures: Computational Studies, Synthesis, and In Vitro Assessment.
J Chem Inf Model
; 62(4): 854-873, 2022 02 28.
Artículo
en Inglés
| MEDLINE | ID: mdl-35143200
2.
HDAC6 as privileged target in drug discovery: A perspective.
Pharmacol Res
; 163: 105274, 2021 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-33171304
3.
Design, synthesis and binding mode of interaction of novel small molecule o-hydroxy benzamides as HDAC3-selective inhibitors with promising antitumor effects in 4T1-Luc breast cancer xenograft model.
Bioorg Chem
; 117: 105446, 2021 12.
Artículo
en Inglés
| MEDLINE | ID: mdl-34717237
4.
Synthesis, biological evaluation, and molecular docking analysis of novel linker-less benzamide based potent and selective HDAC3 inhibitors.
Bioorg Chem
; 114: 105050, 2021 09.
Artículo
en Inglés
| MEDLINE | ID: mdl-34120025
5.
Design, synthesis and biological evaluation of 7-(5-((substituted - amino)-methyl)-thiophen-2-yl)-spiro-[chroman-2,4'-piperidin]-4-one hydrochloride analogues as anticancer agents.
Bioorg Chem
; 112: 104865, 2021 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-33812269
6.
Structure-activity relationship of human carbonic anhydrase-II inhibitors: Detailed insight for future development as anti-glaucoma agents.
Bioorg Chem
; 95: 103557, 2020 01.
Artículo
en Inglés
| MEDLINE | ID: mdl-31911296
7.
Discovery of 1,2,3-triazole based quinoxaline-1,4-di-N-oxide derivatives as potential anti-tubercular agents.
Bioorg Chem
; 100: 103955, 2020 07.
Artículo
en Inglés
| MEDLINE | ID: mdl-32464405
8.
HDAC8 as an emerging target in drug discovery with special emphasis on medicinal chemistry.
Future Med Chem
; 15(10): 885-908, 2023 May.
Artículo
en Inglés
| MEDLINE | ID: mdl-37227732
9.
Selective HDAC3 Inhibitors with Potent In Vivo Antitumor Efficacy against Triple-Negative Breast Cancer.
J Med Chem
; 66(17): 12033-12058, 2023 09 14.
Artículo
en Inglés
| MEDLINE | ID: mdl-37660352
10.
Selective inhibition of histone deacetylase 3 by novel hydrazide based small molecules as therapeutic intervention for the treatment of cancer.
Eur J Med Chem
; 238: 114470, 2022 Aug 05.
Artículo
en Inglés
| MEDLINE | ID: mdl-35635949
11.
Design, synthesis and structure-activity relationship studies of novel spirochromanone hydrochloride analogs as anticancer agents.
Future Med Chem
; 14(5): 325-342, 2022 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-34985322
12.
PT3: A Novel Benzamide Class Histone Deacetylase 3 Inhibitor Improves Learning and Memory in Novel Object Recognition Mouse Model.
ACS Chem Neurosci
; 12(5): 883-892, 2021 03 03.
Artículo
en Inglés
| MEDLINE | ID: mdl-33577290
13.
Design, synthesis and biological evaluation of 1,2,3-triazole based 2-aminobenzimidazoles as novel inhibitors of LasR dependent quorum sensing in Pseudomonas aeruginosa.
RSC Adv
; 9(50): 29273-29292, 2019 Sep 13.
Artículo
en Inglés
| MEDLINE | ID: mdl-35528444
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